日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

M102 activates both NRF2 and HSF1 transcription factor pathways and is neuroprotective in cell and animal models of amyotrophic lateral sclerosis

M102 可激活 NRF2 和 HSF1 转录因子通路,并在肌萎缩侧索硬化症的细胞和动物模型中发挥神经保护作用。

Keerie, Amy F; Martins, Raquel Rua; Allen, Chloe F; Bowden, Katie; Al Mashhadi, Sufana; Marlow, Thomas; Myszczynska, Monika; Thakur, Nikitha; Beal, Selina N; Shaw, Allan; Suresh, Shivani; McKinnon, Scott N; Cooper-Knock, Johnathan; West, Ryan J H; Bonsall, Sam; Daniel, Alex; Wells, Tyler; Kumar, Vedanth; Ellis, Brittany C S; Higgins, Maureen; Dinkova-Kostova, Albena T; Shelkovnikova, Tatyana A; Kalfus, Ira N; Shan, Ning; Shaw, Pamela J; Ferraiuolo, Laura; Mead, Richard J

Tetrazole-containing naphthalene bis-sulfonamide Keap1-Nrf2 interaction inhibitors with unexpected binding modes.

具有意想不到的结合模式的含四唑萘双磺酰胺 Keap1-Nrf2 相互作用抑制剂。

Georgakopoulos Nikolaos D, Talapatra Sandeep K, Dayalan Naidu Sharadha, Dikovskaya Dina, Higgins Maureen, Gatliff Jemma, Nikoloudaki Roxani, Schaap Marjolein, Walker Jasmine M, Wardby Christopher, Dinkova-Kostova Albena T, Harris Sarah, Kozielski Frank, Wells Geoff

Identification of a BACH1 lung cancer signature: A novel tool for understanding BACH1 biology and identifying new inhibitors.

鉴定 BACH1 肺癌特征:了解 BACH1 生物学和鉴定新抑制剂的新工具

Klenja-Skudrinja Donika, Ali Kevin X, Walker David, Higgins Maureen, Patel Angana Ah, Raj Dorota, Creelman Anna, McDowall Charlotte, Taylor Conor, Wenta Tomasz, Larsson Erik, Wiel Clotilde, Sayin Volkan I, de la Vega Laureano

Chalcone constituents pulincisones A-F isolated from Pulicaria incisa with NQO1 inducer activity

从裂叶芍药(Pulicaria incisa)中分离得到的查尔酮成分pulincisones AF具有NQO1诱导活性。

Hamed, Ahmed R; Mohamed, Tarik A; Abdel-Halim, Sally A; El-Razek, Mohamed H Abd; El-Toumy, Sayed A; Higgins, Maureen; Skalicka-Woźniak, Krystyna; Dinkova-Kostova, Albena T; Paré, Paul W; Sakr, Mahmoud M; Hegazy, Mohamed-Elamir F

A fluorescence lifetime-based FLIM-timer for measuring the protein turnover of transcription factor Nrf2 in live cells.

一种基于荧光寿命的 FLIM 计时器,用于测量活细胞中转录因子 Nrf2 的蛋白质周转率

Dikovskaya Dina, Bento-Pereira Claudia, Shiga Kanade, Corno Andrea, Higgins Maureen, Toth Rachel, Saurin Adrian T, Dinkova-Kostova Albena T

Author Correction: Octyl itaconate enhances VSVΔ51 oncolytic virotherapy by multitarget inhibition of antiviral and inflammatory pathways

作者更正:衣康酸辛酯通过多靶点抑制抗病毒和炎症通路增强VSVΔ51溶瘤病毒疗法

Kurmasheva, Naziia; Said, Aida; Wong, Boaz; Kinderman, Priscilla; Han, Xiaoying; Rahimic, Anna H F; Kress, Alena; Carter-Timofte, Madalina E; Holm, Emilia; van der Horst, Demi; Kollmann, Christoph F; Liu, Zhenlong; Wang, Chen; Hoang, Huy-Dung; Kovalenko, Elina; Chrysopoulou, Maria; Twayana, Krishna Sundar; Ottosen, Rasmus N; Svenningsen, Esben B; Begnini, Fabio; Kiib, Anders E; Kromm, Florian E H; Weiss, Hauke J; Di Carlo, Daniele; Muscolini, Michela; Higgins, Maureen; van der Heijden, Mirte; Arulanandam, Rozanne; Bardoul, Angelina; Tong, Tong; Ozsvar, Attila; Hou, Wen-Hsien; Schack, Vivien R; Holm, Christian K; Zheng, Yunan; Ruzek, Melanie; Kalucka, Joanna; de la Vega, Laureano; Elgaher, Walid A M; Korshoej, Anders R; Lin, Rongtuan; Hiscott, John; Poulsen, Thomas B; O'Neill, Luke A; Roy, Dominic G; Rinschen, Markus M; van Montfoort, Nadine; Diallo, Jean-Simon; Farin, Henner F; Alain, Tommy; Olagnier, David

Publisher Correction: A DHODH inhibitor increases p53 synthesis and enhances tumor cell killing by p53 degradation blockage

出版商更正:DHODH抑制剂通过阻断p53降解来增加p53合成并增强肿瘤细胞杀伤作用。

Ladds, Marcus J G W; van Leeuwen, Ingeborg M M; Drummond, Catherine J; Chu, Su; Healy, Alan R; Popova, Gergana; Fernández, Andrés Pastor; Mollick, Tanzina; Darekar, Suhas; Sedimbi, Saikiran K; Nekulova, Marta; Sachweh, Marijke C C; Campbell, Johanna; Higgins, Maureen; Tuck, Chloe; Popa, Mihaela; Safont, Mireia Mayoral; Gelebart, Pascal; Fandalyuk, Zinayida; Thompson, Alastair M; Svensson, Richard; Gustavsson, Anna-Lena; Johansson, Lars; Färnegårdh, Katarina; Yngve, Ulrika; Saleh, Aljona; Haraldsson, Martin; D'Hollander, Agathe C A; Franco, Marcela; Zhao, Yan; Håkansson, Maria; Walse, Björn; Larsson, Karin; Peat, Emma M; Pelechano, Vicent; Lunec, John; Vojtesek, Borivoj; Carmena, Mar; Earnshaw, William C; McCarthy, Anna R; Westwood, Nicholas J; Arsenian-Henriksson, Marie; Lane, David P; Bhatia, Ravi; McCormack, Emmet; Laín, Sonia

Pirin, an Nrf2-Regulated Protein, Is Overexpressed in Human Colorectal Tumors

Pirin是一种受Nrf2调控的蛋白质,在人类结直肠肿瘤中过度表达。

Zhang, Ying; Knatko, Elena V; Higgins, Maureen; Dayalan Naidu, Sharadha; Smith, Gillian; Honda, Tadashi; de la Vega, Laureano; Dinkova-Kostova, Albena T

Nrf2 activation does not affect adenoma development in a mouse model of colorectal cancer

在小鼠结直肠癌模型中,Nrf2激活不影响腺瘤的发生发展。

Knatko, Elena V; Castro, Cecilia; Higgins, Maureen; Zhang, Ying; Honda, Tadashi; Henderson, Colin J; Wolf, C Roland; Griffin, Julian L; Dinkova-Kostova, Albena T

Publisher Correction: A DHODH inhibitor increases p53 synthesis and enhances tumor cell killing by p53 degradation blockage

出版商更正:DHODH抑制剂通过阻断p53降解来增加p53合成并增强肿瘤细胞杀伤作用。

Ladds, Marcus J G W; van Leeuwen, Ingeborg M M; Drummond, Catherine J; Chu, Su; Healy, Alan R; Popova, Gergana; Pastor Fernández, Andrés; Mollick, Tanzina; Darekar, Suhas; Sedimbi, Saikiran K; Nekulova, Marta; Sachweh, Marijke C C; Campbell, Johanna; Higgins, Maureen; Tuck, Chloe; Popa, Mihaela; Safont, Mireia Mayoral; Gelebart, Pascal; Fandalyuk, Zinayida; Thompson, Alastair M; Svensson, Richard; Gustavsson, Anna-Lena; Johansson, Lars; Färnegårdh, Katarina; Yngve, Ulrika; Saleh, Aljona; Haraldsson, Martin; D'Hollander, Agathe C A; Franco, Marcela; Zhao, Yan; Håkansson, Maria; Walse, Björn; Larsson, Karin; Peat, Emma M; Pelechano, Vicent; Lunec, John; Vojtesek, Borivoj; Carmena, Mar; Earnshaw, William C; McCarthy, Anna R; Westwood, Nicholas J; Arsenian-Henriksson, Marie; Lane, David P; Bhatia, Ravi; McCormack, Emmet; Laín, Sonia