Selective covalent targeting of GPX4 using masked nitrile-oxide electrophiles
使用掩蔽的腈氧化物亲电试剂对 GPX4 进行选择性共价靶向
期刊:Nature Chemical Biology
影响因子:12.9
doi:10.1038/s41589-020-0501-5
John K Eaton, Laura Furst, Richard A Ruberto, Dieter Moosmayer, André Hilpmann, Matthew J Ryan, Katja Zimmermann, Luke L Cai, Michael Niehues, Volker Badock, Anneke Kramm, Sixun Chen, Roman C Hillig, Paul A Clemons, Stefan Gradl, Claire Montagnon, Kiel E Lazarski, Sven Christian, Besnik Bajrami, Rol