日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Capsaicin-Inspired Hydroxamate Hybrids as Selective HDAC6 Inhibitors with Antiproliferative Activity in Hematological Malignancies

辣椒素衍生的羟肟酸酯杂合物作为选择性 HDAC6 抑制剂,在血液恶性肿瘤中具有抗增殖活性

Gimenez Borges, Lara; Alves, Thais Nascimento de Oliveira; Vassiliades, Sandra Valeria; Carlos, Jorge Antonio Elias Godoy; Waitman, Karoline de Barros; Hilscher, Sebastian; Schutkowski, Mike; Sippl, Wolfgang; Tavares, Maurício Temotheo; Toledo, Monica Franco Zannini Junqueira; Costa-Lotufo, Letícia Veras; Kronenberger, Thales; Machado-Neto, João Agostinho; Parise-Filho, Roberto

The protein deacetylase HDAC10 controls DNA replication in malignant lymphoid cells

蛋白质去乙酰化酶HDAC10控制恶性淋巴细胞中的DNA复制。

Mieland, Andreas O; Petrosino, Giuseppe; Dejung, Mario; Chen, Jia-Xuan; Fulzele, Amitkumar; Mahmoudi, Fereshteh; Tu, Jia-Wey; Mustafa, Al-Hassan M; Zeyn, Yanira; Hieber, Christoph; Bros, Matthias; Schnöder, Tina M; Heidel, Florian H; Najafi, Sara; Oehme, Ina; Hofmann, Ilse; Schutkowski, Mike; Hilscher, Sebastian; Kosan, Christian; Butter, Falk; Bhatia, Sanil; Sippl, Wolfgang; Krämer, Oliver H

Dona Flor and her two husbands: Discovery of novel HDAC6/AKT2 inhibitors for myeloid cancer treatment

唐娜·弗洛尔和她的两位丈夫:发现用于治疗髓系癌症的新型HDAC6/AKT2抑制剂

Waitman, Karoline B; Martin, Holli-Joi; Carlos, Jorge A E G; Braga, Rodolpho C; Souza, Vinícius A M; Melo-Filho, Cleber C; Hilscher, Sebastian; Toledo, Mônica F Z J; Tavares, Maurício T; Costa-Lotufo, Letícia V; Machado-Neto, João A; Schutkowski, Mike; Sippl, Wolfgang; Kronenberger, Thales; Alves, Vinicius M; Parise-Filho, Roberto; Muratov, Eugene N

Substrate-Guided Development of HDAC11-Selective Inhibitors Featuring α‑Amino Amide Zinc-Binding Groups

基于底物导向的HDAC11选择性抑制剂的开发,该抑制剂具有α-氨基酰胺锌结合基团

Hilscher, Sebastian; Meleshin, Marat; Baselious, Fady; Barinka, Cyril; Sippl, Wolfgang; Schutkowski, Mike; Schiene-Fischer, Cordelia

Development of potent and selective tetrahydro-β-carboline-based HDAC6 inhibitors with promising activity against triple-negative breast cancer.

开发高效且选择性的四氢-β-咔啉类HDAC6抑制剂,对三阴性乳腺癌具有良好的活性

Fathy Aya, Allam Amro, ElHady Ahmed K, El-Gamil Dalia S, Lin Kai-Chun, Chang Yen-Hua, Lee Yu-Hsuan, Hilscher Sebastian, Schutkowski Mike, Ibrahim Hany S, Chen Shun-Hua, Chen Chun-Hong, Abadi Ashraf H, Sippl Wolfgang, Chen Po-Jen, Cheng Yi-Sheng, Abdel-Halim Mohammad

Comparative Structure-Based Virtual Screening Utilizing Optimized AlphaFold Model Identifies Selective HDAC11 Inhibitor

利用优化的AlphaFold模型进行基于结构的比较虚拟筛选,鉴定出选择性HDAC11抑制剂

Baselious, Fady; Hilscher, Sebastian; Robaa, Dina; Barinka, Cyril; Schutkowski, Mike; Sippl, Wolfgang