日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CSN5i-3 is an orthosteric molecular glue inhibitor of COP9 signalosome

CSN5i-3 是一种 COP9 信号体的正构分子胶抑制剂。

Shi, Huigang; Wang, Xiaorong; Yu, Clinton; Mao, Haibin; Jiao, Fenglong; Braitbard, Merav; Shor, Ben; Zhang, Zhongsheng; Hinds, Thomas R; Cao, Shiyun; Fan, Erkang; Schneidman-Duhovny, Dina; Huang, Lan; Zheng, Ning

Orthosteric Molecular Glue Inhibits COP9 Signalosome with Substrate-Dependent Potency

正构分子胶抑制COP9信号复合物的效力取决于底物

Shi, Huigang; Wang, Xiaorong; Yu, Clinton; Mao, Haibin; Jiao, Fenglong; Braitbard, Merav; Shor, Ben; Zhang, Zhongsheng; Hinds, Thomas R; Cao, Shiyun; Fan, Erkang; Schneidman-Duhovny, Dina; Huang, Lan; Zheng, Ning

Structural insights into DDA1 function as a core component of the CRL4-DDB1 ubiquitin ligase

对DDA1作为CRL4-DDB1泛素连接酶核心组分的功能进行结构解析

Shabek, Nitzan; Ruble, James; Waston, Claire J; Garbutt, Kenneth C; Hinds, Thomas R; Li, Ti; Zheng, Ning

Enzyme assays for cGMP hydrolyzing phosphodiesterases

cGMP水解磷酸二酯酶的酶活性测定

Rybalkin, Sergei D; Hinds, Thomas R; Beavo, Joseph A

Kaempferia parviflora, a plant used in traditional medicine to enhance sexual performance contains large amounts of low affinity PDE5 inhibitors.

姜黄(Kaempferia parviflora)是一种在传统医学中用于增强性功能的植物,含有大量低亲和力 PDE5 抑制剂

Temkitthawon Prapapan, Hinds Thomas R, Beavo Joseph A, Viyoch Jarupa, Suwanborirux Khanit, Pongamornkul Wittaya, Sawasdee Pattara, Ingkaninan Kornkanok

Characterization of a novel cAMP-binding, cAMP-specific cyclic nucleotide phosphodiesterase (TcrPDEB1) from Trypanosoma cruzi.

对克氏锥虫中一种新型 cAMP 结合、cAMP 特异性环核苷酸磷酸二酯酶 (TcrPDEB1) 进行表征

Díaz-Benjumea Rocío, Laxman Sunil, Hinds Thomas R, Beavo Joseph A, Rascón Ana