日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

SHP2 Inhibition Sensitizes Diverse Oncogene-Addicted Solid Tumors to Re-treatment with Targeted Therapy

SHP2 抑制可增强多种致癌基因依赖性实体肿瘤对靶向治疗的再治疗敏感性

Alexander Drilon, Manish R Sharma #, Melissa L Johnson #, Timothy A Yap #, Shirish Gadgeel, Dale Nepert, Gang Feng, Micaela B Reddy, Allison S Harney, Mohamed Elsayed, Adam W Cook, Christina E Wong, Ronald J Hinklin, Yutong Jiang, Eric N Brown, Nickolas A Neitzel, Ellen R Laird, Wen-I Wu, Anurag Sin

5-Alkyl-2-urea-Substituted Pyridines: Identification of Efficacious Glucokinase Activators with Improved Properties

5-烷基-2-脲取代的吡啶:高效葡萄糖激酶激活剂及其性能的改进

Kohn, Todd J; Du, Xiaohui; Lai, SuJen; Xiong, YuMei; Komorowski, Renee; Veniant, Murielle; Fu, Zice; Jiao, Xianyun; Pattaropong, Vatee; Chow, David; Cardozo, Mario; Jin, Lixia; Conn, Marion; DeWolf, Walter E Jr; Kraser, Christopher F; Hinklin, Ronald J; Boys, Mark L; Medina, Julio C; Houze, Jonathan; Dransfield, Paul; Coward, Peter

Novel Series of Potent Glucokinase Activators Leading to the Discovery of AM-2394

新型强效葡萄糖激酶激活剂系列研究促成了AM-2394的发现

Dransfield, Paul J; Pattaropong, Vatee; Lai, Sujen; Fu, Zice; Kohn, Todd J; Du, Xiaohui; Cheng, Alan; Xiong, Yumei; Komorowski, Renee; Jin, Lixia; Conn, Marion; Tien, Eric; DeWolf, Walter E Jr; Hinklin, Ronald J; Aicher, Thomas D; Kraser, Christopher F; Boyd, Steven A; Voegtli, Walter C; Condroski, Kevin R; Veniant-Ellison, Murielle; Medina, Julio C; Houze, Jonathan; Coward, Peter

C5-Alkyl-2-methylurea-Substituted Pyridines as a New Class of Glucokinase Activators

C5-烷基-2-甲基脲取代的吡啶类化合物作为一类新型葡萄糖激酶激活剂

Du, Xiaohui; Hinklin, Ronald J; Xiong, Yumei; Dransfield, Paul; Park, Jaehyeon; Kohn, Todd J; Pattaropong, Vatee; Lai, SuJen; Fu, Zice; Jiao, Xianyun; Chow, David; Jin, Lixia; Davda, Jasmine; Veniant, Murielle M; Anderson, Deborah A; Baer, Brian R; Bencsik, Josef R; Boyd, Steven A; Chicarelli, Mark Joseph; Mohr, Peter J; Wang, Bin; Condroski, Kevin R; DeWolf, Walter E; Conn, Marion; Tran, Thanhvien; Yang, Jerry; Aicher, Thomas D; Medina, Julio C; Coward, Peter; Houze, Jonathan B

Primary xenografts of human prostate tissue as a model to study angiogenesis induced by reactive stroma

以人前列腺组织原代异种移植为模型,研究反应性基质诱导的血管生成

Montecinos, Viviana P; Godoy, Alejandro; Hinklin, Jennifer; Vethanayagam, R Robert; Smith, Gary J