Translational Preclinical PET Imaging and Metabolic Evaluation of a New Cannabinoid 2 Receptor (CB(2)R) Radioligand, (Z)-N-(3-(2-(2-[(18)F]Fluoroethoxy)ethyl)-4,5-dimethylthiazol-2(3H)-ylidene)-2,2,3,3-tetramethylcyclopropane-1-carboxamide
一种新型大麻素2受体(CB(2)R)放射性配体(Z)-N-(3-(2-(2-[(18)F]氟乙氧基)乙基)-4,5-二甲基噻唑-2(3H)-亚基)-2,2,3,3-四甲基环丙烷-1-甲酰胺的转化临床前PET成像和代谢评价
期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.4c00348
Auvity, Sylvain; Attili, Bala; Caillé, Fabien; Goislard, Maud; Cayla, Jérôme; Hinnen, Françoise; Demphel, Stéphane; Brulon, Vincent; Bottlaender, Michel; Leroy, Claire; Bormans, Guy; Kuhnast, Bertrand; Peyronneau, Marie-Anne