日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Effects of novel TRPA1 receptor agonist ASP7663 in models of drug-induced constipation and visceral pain

新型 TRPA1 受体激动剂 ASP7663 对药物性便秘和内脏痛模型的影响

Ryosuke Kojima, Katsura Nozawa, Hitoshi Doihara, Yoshihiro Keto, Hidetaka Kaku, Toshihide Yokoyama, Hiroyuki Itou

A novel glycine transporter-1 (GlyT1) inhibitor, ASP2535 (4-[3-isopropyl-5-(6-phenyl-3-pyridyl)-4H-1,2,4-triazol-4-yl]-2,1,3-benzoxadiazole), improves cognition in animal models of cognitive impairment in schizophrenia and Alzheimer's disease

一种新型甘氨酸转运蛋白-1 (GlyT1) 抑制剂 ASP2535(4-[3-异丙基-5-(6-苯基-3-吡啶基)-4H-1,2,4-三唑-4-基]-2,1,3-苯并恶二唑)可改善精神分裂症和阿尔茨海默病认知障碍动物模型的认知能力

Katsuya Harada, Kazuhiro Nakato, Junko Yarimizu, Mayako Yamazaki, Masahiko Morita, Shinji Takahashi, Masaki Aota, Kyoko Saita, Hitoshi Doihara, Yuichiro Sato, Takayuki Yamaji, Keni Ni, Nobuya Matsuoka

TRPA1 regulates gastrointestinal motility through serotonin release from enterochromaffin cells

TRPA1 通过肠嗜铬细胞释放血清素来调节胃肠运动

Katsura Nozawa, Eri Kawabata-Shoda, Hitoshi Doihara, Ryosuke Kojima, Hidetsugu Okada, Shinobu Mochizuki, Yorikata Sano, Kohei Inamura, Hitoshi Matsushime, Tomonobu Koizumi, Toshihide Yokoyama, Hiroyuki Ito