日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Potent and Efficacious Influenza PB2 Inhibitors

发现高效强效的流感病毒PB2抑制剂

Wu, Jun; Liu, Yongfu; Li, Dongbo; Wang, Lisha; Neidhart, Werner; Chen, Bo; Hochstrasser, Remo; Kuglstatter, Andreas; Gasser, Rodolfo; Qiu, Hongxia; Shi, Tianlai; Chao, Suzan Keen; Gao, Junjun; Shen, Hong C; Tan, Xuefei

A Highly Selective and Versatile Probe Platform for Visualization of Monoacylglycerol Lipase

一种用于可视化单酰甘油脂肪酶的高选择性和多功能探针平台

Hentsch, Axel; Guberman, Mónica; Radetzki, Silke; Kaushik, Sofia; Huizenga, Mirjam; Paul, Jerome; Schippers, Maria; Benz, Jörg; Kuhn, Bernd; Heer, Dominik; Topp, Andreas; Esteves Gloria, Ludivine; Walter, Alexander; Hochstrasser, Remo; Wittwer, Matthias B; von Kries, Jens Peter; Collin, Ludovic; Blaising, Julie; van der Stelt, Mario; Lipstein, Noa; Grether, Uwe; Nazaré, Marc

Expediting hit-to-lead progression in drug discovery through reaction prediction and multi-dimensional optimization

通过反应预测和多维优化加速药物发现中的先导化合物转化进程

Nippa, David F; Atz, Kenneth; Stenzhorn, Yannick; Müller, Alex T; Tosstorff, Andreas; Benz, Jörg; Binch, Hayley; Bürkler, Markus; Haider, Achi; Heer, Dominik; Hochstrasser, Remo; Kramer, Christian; Reutlinger, Michael; Schneider, Petra; Shema, Thierry; Topp, Andreas; Walter, Alexander; Wittwer, Matthias B; Wolfard, Jens; Kuhn, Bernd; van der Stelt, Mario; Martin, Rainer E; Grether, Uwe; Schneider, Gisbert

Highly Specific Miniaturized Fluorescent Monoacylglycerol Lipase Probes Enable Translational Research

高特异性微型荧光单酰甘油脂肪酶探针助力转化研究

Hentsch, Axel; Guberman, Mónica; Radetzki, Silke; Kaushik, Sofia; Huizenga, Mirjam; He, Yingfang; Contzen, Jörg; Kuhn, Bernd; Benz, Jörg; Schippers, Maria; Paul, Jerome; Leibrock, Lea; Collin, Ludovic; Wittwer, Matthias; Topp, Andreas; O'Hara, Fionn; Heer, Dominik; Hochstrasser, Remo; Blaising, Julie; von Kries, Jens P; Mu, Linjing; van der Stelt, Mario; Mergenthaler, Philipp; Lipstein, Noa; Grether, Uwe; Nazaré, Marc

CellEKT: A Robust Chemical Proteomics Workflow to Profile Cellular Target Engagement of Kinase Inhibitors.

CellEKT:一种稳健的化学蛋白质组学工作流程,用于分析激酶抑制剂的细胞靶标结合情况

Rüegger Joel, Gagestein Berend, Janssen Antonius P A, Valeanu Alexandra, Mori Alger Lazo, van der Peet Marielle, Boutkan Michael S, Florea Bogdan I, Henneman Alex A, Hochstrasser Remo, Wang Haiyan, Westwood Paul, Topp Andreas, Gomez Barila Patricia M, Medema Jan Paul, Jimenez Connie R, Woersdoerfer Bigna, Kirchner Stephan, Zhang Jitao David, Grether Uwe, Rufer Arne C, van der Stelt Mario