The Pan-RAF-MEK Nondegrading Molecular Glue NST-628 Is a Potent and Brain-Penetrant Inhibitor of the RAS-MAPK Pathway with Activity across Diverse RAS- and RAF-Driven Cancers
泛 RAF-MEK 非降解分子胶 NST-628 是一种强效的脑渗透性 RAS-MAPK 通路抑制剂,可有效治疗多种 RAS 和 RAF 驱动的癌症
期刊:Cancer Discovery
影响因子:29.7
doi:10.1158/2159-8290.CD-24-0139
Meagan B Ryan #, Bradley Quade #, Natasha Schenk, Zhong Fang, Marshall Zingg, Steven E Cohen, Brooke M Swalm, Chun Li, Ayşegül Özen, Chaoyang Ye, Maria Stella Ritorto, Xin Huang, Arvin C Dar, Yongxin Han, Klaus P Hoeflich, Michael Hale, Margit Hagel