日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

RETRACTED: Naamneh et al. Structure-Activity Relationship of Synthetic Linear KTS-Peptides Containing Meta-Aminobenzoic Acid as Antagonists of α1β1 Integrin with Anti-Angiogenic and Melanoma Anti-Tumor Activities. Pharmaceuticals 2024, 17, 549

撤稿:Naamneh 等人,《含间氨基苯甲酸的合成线性 KTS 肽作为 α1β1 整合素拮抗剂的构效关系及其抗血管生成和抗黑色素瘤活性》,Pharmaceuticals 2024, 17, 549

Naamneh, Majdi Saleem; Momic, Tatjana; Klazas, Michal; Grosche, Julius; Eble, Johannes A; Marcinkiewicz, Cezary; Khazanov, Netaly; Senderowitz, Hanoch; Hoffman, Amnon; Gilon, Chaim; Katzhendler, Jehoshua; Lazarovici, Philip

Development of Clarstatin, a Novel Drug Lead for the Therapy of Autoimmune Uveitis

克拉司他汀(Clarstatin)的研发:一种用于治疗自身免疫性葡萄膜炎的新型先导药物

Merzbach, Shira; Hoffman, Amnon; Lazarovici, Philip; Gilon, Chaim; Amer, Radgonde

The Synthesis of SNAC Phenolate Salts and the Effect on Oral Bioavailability of Semaglutide

SNAC酚盐的合成及其对司美格鲁肽口服生物利用度的影响

Shapira-Furman, Tovi; Bar-Hai, Ayala; Hoffman, Amnon; Domb, Abraham J

Treatment with αvβ3-integrin-specific 29P attenuates pressure-overload induced cardiac remodelling after transverse aortic constriction in mice

在小鼠中,用αvβ3整合素特异性29P治疗可减轻横向主动脉缩窄后压力超负荷诱导的心脏重塑。

Njegić, Alexandra; Laid, Lina; Zi, Min; Maniati, Eleni; Wang, Jun; Chelu, Alexandru; Wisniewski, Laura; Hunter, Jenna; Prehar, Sukhpal; Stafford, Nicholas; Gilon, Chaim; Hoffman, Amnon; Weinmüller, Michael; Kessler, Horst; Cartwright, Elizabeth J; Hodivala-Dilke, Kairbaan

Cyclizing Painkillers: Development of Backbone-Cyclic TAPS Analogs

环状止痛药:主链环状TAPS类似物的开发

Talhami, Alaa; Swed, Avi; Hess, Shmuel; Ovadia, Oded; Greenberg, Sarit; Schumacher-Klinger, Adi; Rosenthal, David; Shalev, Deborah E; Hurevich, Mattan; Lazarovici, Philip; Hoffman, Amnon; Gilon, Chaim

Development of a Novel Backbone Cyclic Peptide Inhibitor of the Innate Immune TLR/IL1R Signaling Protein MyD88.

开发一种新型的先天免疫 TLR/IL1R 信号蛋白 MyD88 骨架环肽抑制剂

Dishon Shira, Schumacher Adi, Fanous Joseph, Talhami Alaa, Kassis Ibrahim, Karussis Dimitrios, Gilon Chaim, Hoffman Amnon, Nussbaum Gabriel

Antihyperglycaemic activity of 2,4:3,5-dibenzylidene-D-xylose-diethyl dithioacetal in diabetic mice

2,4:3,5-二亚苄基-D-木糖-二乙基二硫缩醛在糖尿病小鼠中的降血糖活性

Gruzman, Arie; Elgart, Anna; Viskind, Olga; Billauer, Hana; Dotan, Sharon; Cohen, Guy; Mishani, Eyal; Hoffman, Amnon; Cerasi, Erol; Sasson, Shlomo

Developing potent backbone cyclic peptides bearing the shared epitope sequence as rheumatoid arthritis drug-leads

开发具有共同表位序列的强效骨架环肽作为类风湿性关节炎先导药物

Naveh, Shirly; Tal-Gan, Yftah; Ling, Song; Hoffman, Amnon; Holoshitz, Joseph; Gilon, Chaim

Structure-activity relationship and metabolic stability studies of backbone cyclization and N-methylation of melanocortin peptides

黑皮质素肽骨架环化和N-甲基化的构效关系及代谢稳定性研究

Linde, Yaniv; Ovadia, Oded; Safrai, Eli; Xiang, Zhimin; Portillo, Federico P; Shalev, Deborah E; Haskell-Luevano, Carrie; Hoffman, Amnon; Gilon, Chaim

DP-155, a lecithin derivative of indomethacin, is a novel nonsteroidal antiinflammatory drug for analgesia and Alzheimer's disease therapy

DP-155是吲哚美辛的卵磷脂衍生物,是一种新型非甾体类抗炎药,可用于镇痛和治疗阿尔茨海默病。

Dvir, Eran; Elman, Anat; Simmons, Danielle; Shapiro, Israel; Duvdevani, Revital; Dahan, Arik; Hoffman, Amnon; Friedman, Jonathan E