Camostat mesylate inhibits SARS-CoV-2 activation by TMPRSS2-related proteases and its metabolite GBPA exerts antiviral activity
甲磺酸卡莫司他可抑制TMPRSS2相关蛋白酶对SARS-CoV-2的激活,其代谢产物GBPA具有抗病毒活性。
期刊:EBioMedicine
影响因子:10.8
doi:10.1016/j.ebiom.2021.103255
Hoffmann, Markus; Hofmann-Winkler, Heike; Smith, Joan C; Krüger, Nadine; Arora, Prerna; Sørensen, Lambert K; Søgaard, Ole S; Hasselstrøm, Jørgen Bo; Winkler, Michael; Hempel, Tim; Raich, Lluís; Olsson, Simon; Danov, Olga; Jonigk, Danny; Yamazoe, Takashi; Yamatsuta, Katsura; Mizuno, Hirotaka; Ludwig, Stephan; Noé, Frank; Kjolby, Mads; Braun, Armin; Sheltzer, Jason M; Pöhlmann, Stefan