日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of Derivatives of the Antibiotic Albicidin: The N-Terminal Fragment as Key to Control Potency and Resistance Mediated by the Binding Protein AlbA

抗生素白菌素衍生物的合成:N端片段是控制其效力和耐药性的关键,而耐药性是由结合蛋白AlbA介导的。

Kulike-Koczula, Marcel; Hommernick, Kay; Ghimire, Leela B; Kosol, Simone; Zborovsky, Lieby; Seidel, Maria; Sattler, Nicole; Mainz, Andi; Weston, John B; Ghilarov, Dmitry; Süssmuth, Roderich D

Molecular mechanism of topoisomerase poisoning by the peptide antibiotic albicidin

肽类抗生素白菌素对拓扑异构酶的毒害分子机制

Michalczyk, Elizabeth; Hommernick, Kay; Behroz, Iraj; Kulike, Marcel; Pakosz-Stępień, Zuzanna; Mazurek, Lukasz; Seidel, Maria; Kunert, Maria; Santos, Karine; von Moeller, Holger; Loll, Bernhard; Weston, John B; Mainz, Andi; Heddle, Jonathan G; Süssmuth, Roderich D; Ghilarov, Dmitry

Transcription activation by the resistance protein AlbA as a tool to evaluate derivatives of the antibiotic albicidin

利用抗性蛋白AlbA的转录激活作用来评价抗生素白菌素衍生物

Kosol, Simone; Rostock, Lida; Barsig, Jonas; Tabarelli, Theresa; Hommernick, Kay; Kulike, Marcel; Eulberg, Tobias; Seidel, Maria; Behroz, Iraj; Kleebauer, Leonardo; Grätz, Stefan; Mainz, Andi; Süssmuth, Roderich D

Acetylenic Replacement of Albicidin's Methacrylamide Residue Circumvents Detrimental E/Z Photoisomerization and Preserves Antibacterial Activity

用乙炔基取代白菌素中的甲基丙烯酰胺残基可避免有害的E/Z光异构化并保持其抗菌活性。

Behroz, Iraj; Kleebauer, Leonardo; Hommernick, Kay; Seidel, Maria; Grätz, Stefan; Mainz, Andi; Weston, John B; Süssmuth, Roderich D