日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural basis of THC analog activity at the Cannabinoid 1 receptor.

THC类似物在大麻素1受体上的活性结构基础

Thorsen Thor S, Kulkarni Yashraj, Sykes David A, Bøggild Andreas, Drace Taner, Hompluem Pattarin, Iliopoulos-Tsoutsouvas Christos, Nikas Spyros P, Daver Henrik, Makriyannis Alexandros, Nissen Poul, Gajhede Michael, Veprintsev Dmitry B, Boesen Thomas, Kastrup Jette S, Gloriam David E

Combined docking and machine learning identify key molecular determinants of ligand pharmacological activity on β2 adrenoceptor

结合分子对接和机器学习技术,识别出配体对β2肾上腺素受体药理活性的关键分子决定因素

Jiménez-Rosés, Mireia; Morgan, Bradley Angus; Jimenez Sigstad, Maria; Tran, Thuy Duong Zoe; Srivastava, Rohini; Bunsuz, Asuman; Borrega-Román, Leire; Hompluem, Pattarin; Cullum, Sean A; Harwood, Clare R; Koers, Eline J; Sykes, David A; Styles, Iain B; Veprintsev, Dmitry B