日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Combinations of the azaquinazoline anti-Wolbachia agent, AWZ1066S, with benzimidazole anthelmintics synergise to mediate sub-seven-day sterilising and curative efficacies in experimental models of filariasis

抗沃尔巴克氏体药物AWZ1066S(一种氮杂喹唑啉类药物)与苯并咪唑类驱虫药联合使用,可产生协同作用,在丝虫病实验模型中于7天内达到灭菌和治愈效果。

Hegde, Shrilakshmi; Marriott, Amy E; Pionnier, Nicolas; Steven, Andrew; Bulman, Christina; Gunderson, Emma; Vogel, Ian; Koschel, Marianne; Ehrens, Alexandra; Lustigman, Sara; Voronin, Denis; Tricoche, Nancy; Hoerauf, Achim; Hübner, Marc P; Sakanari, Judy; Aljayyoussi, Ghaith; Gusovsky, Fabian; Dagley, Jessica; Hong, David W; O'Neill, Paul; Ward, Steven A; Taylor, Mark J; Turner, Joseph D

Heterocyclic amines reduce insulin-induced AKT phosphorylation and induce gluconeogenic gene expression in human hepatocytes

杂环胺降低胰岛素诱导的 AKT 磷酸化并诱导人类肝细胞中的糖异生基因表达

Kennedy M Walls, Kyung U Hong, David W Hein

Generation of quinolone antimalarials targeting the Plasmodium falciparum mitochondrial respiratory chain for the treatment and prophylaxis of malaria.

开发针对恶性疟原虫线粒体呼吸链的喹诺酮类抗疟药,用于治疗和预防疟疾

Biagini Giancarlo A, Fisher Nicholas, Shone Alison E, Mubaraki Murad A, Srivastava Abhishek, Hill Alisdair, Antoine Thomas, Warman Ashley J, Davies Jill, Pidathala Chandrakala, Amewu Richard K, Leung Suet C, Sharma Raman, Gibbons Peter, Hong David W, Pacorel Bénédicte, Lawrenson Alexandre S, Charoensutthivarakul Sitthivut, Taylor Lee, Berger Olivier, Mbekeani Alison, Stocks Paul A, Nixon Gemma L, Chadwick James, Hemingway Janet, Delves Michael J, Sinden Robert E, Zeeman Anne-Marie, Kocken Clemens H M, Berry Neil G, O'Neill Paul M, Ward Stephen A

Identification of novel antimalarial chemotypes via chemoinformatic compound selection methods for a high-throughput screening program against the novel malarial target, PfNDH2: increasing hit rate via virtual screening methods.

通过化学信息学化合物选择方法鉴定新型抗疟疾化学类型,用于针对新型疟疾靶点 PfNDH2 的高通量筛选程序:通过虚拟筛选方法提高命中率

Sharma Raman, Lawrenson Alexandre S, Fisher Nicholas E, Warman Ashley J, Shone Alison E, Hill Alasdair, Mbekeani Alison, Pidathala Chandrakala, Amewu Richard K, Leung Suet, Gibbons Peter, Hong David W, Stocks Paul, Nixon Gemma L, Chadwick James, Shearer Joanne, Gowers Ian, Cronk David, Parel Serge P, O'Neill Paul M, Ward Stephen A, Biagini Giancarlo A, Berry Neil G

Modeling the trade-off between effective case management and imported malaria cases in different settings of P. falciparum malaria transmission intensity

在不同恶性疟原虫疟疾传播强度环境下,建立有效病例管理与输入性疟疾病例之间权衡模型

Billingsley, Peter F; Storm, Janet; Müller, Sylke; Batwala, Vincent; Magnussen, Pascal; Nuwaha, Fred; Dahlbäck, Madeleine; Jørgensen, Lars M; Christoffersen, Stig; Nielsen, Morten A; Theander, Thor G; Arnot, David E; Larsen, Sine; Salanti, Ali; Sibley, Carol Hopkins; Liu, Weimin; Li, Yingying; Learn, Gerald H; Rudicell, Rebecca S; Robertson, Joel D; Keele, Brandon F; Ndjango, Jean-Bosco N; Sanz, Crickette M; Morgan, David B; Locatelli, Sabrina; Gonder, Mary K; Kranzusch, Philip J; Walsh, Peter D; Delaporte, Eric; Mpoudi-Ngole, Eitel; Georgiev, Alexander V; Muller, Martin N; Shaw, George M; Peeters, Martine; Sharp, Paul M; Rayner, Julian C; Hahn, Beatrice H; Deplaine, Guillaume; Safeukui, Innocent; Jeddi, Fakhri; Lacoste, François; Brousse, Valentine; Perrot, Sylvie; Biligui, Sylvestre; Guillotte, Micheline; Guitton, Corinne; Dokmak, Safi; Aussilhou, Béatrice; Sauvanet, Alain; Couvelard, Anne; Paye, François; Thellier, Marc; Mazier, Dominique; Milon, Geneviève; Mohandas, Narla; Puijalon, Odile Mercereau; David, Peter H; Buffet, Pierre A; Di Pasquale, Aurelio; Maire, Nicolas; Smith, Thomas; Jean-Bernard, Duchemin; Cyrille, Czeher; Rabiou, Labbo; Lamine, Ibrahim M; Stefan, Hoyer; Isabelle, Jeanne; Maude, Richard James; Sayeed, Abdullah Abu; Beare, Nicholas AV; Charunwatthana, Prakaykaew; Faiz, Abul M; Hossain, Amir; Yunus, Emran Bin; Hoque, Gofranul M; Hasan, Mahtab Uddin; White, Nicholas J; Day, Nicholas PJ; Dondorp, Arjen M; Mota, Maria M; Staines, Henry; Assogba, Benoît S; Djogbenou, Luc S; Dabiré, Roch K; Diabaté, Abdoulaye; Baldet, Thierry; Fatih, Farrah A; Siner, Angela; Ahmed, Atique; Woon, Lu Chan; Craig, Alister; Staines, Henry M; Singh, Balbir; Krishna, Sanjeev; Cox-Singh, Janet; Felger, Ingrid; Schoepflin, Sonja; Kiniboro, Benson; Zimmerman, Peter A; Mueller, Ivo; Gholizadeh, Saber; Karimi, Ameneh; Bayat, Nooshin; Djadid, Navid Dinparast; Zakeri, Sedigheh; Rodrigues, Louise A; Henriques, Gisela; Borges, Sofia T; Hunt, Paul; Sanchez, Cecília P; Martinelli, Axel; Cravo, Pedro; Martins, Joao; Zwi, Anthony; Kelly, Paul; Niemand, J; Birkholtz, L; Louw, AI; Kirk, K; Riglar, David; Richard, Dave; Boyle, Michelle; Wilson, Danny; Angrisano, Fiona; Turnbull, Lynne; Whitchurch, Cynthia; Cowman, Alan; Beeson, James; Ralph, Stuart; Baum, Jake; Kapulu, Melissa C; Biswas, Sumi; Blagborough, Andrew; Gilbert, Sarah C; Sinden, Robert E; Hill, Adrian VS; Jones, Matthew L; Collins, Mark O; Choudhary, Jyoti; Rayner, Julian C; Kaiser, Marco; Bray, Dorothy H; Zommers, Zinta; Couacy-Hymann, Emmanuel; Gillespie, Thomas R; Ellerbrok, Heinz; Leendertz, Fabian H; Gouagna, Louis C; Bancone, Germana; Yao, Frank; Costantini, Carlo; Ouedraogo, Jean-Bosco; Modiano, David; Hulden, Lena; Tanabe, Kazuyuki; Mita, Toshihiro; Balloux, Francois; Saeed, Sadia; Tremp, Annie Z; Dessens, Johannes T; Skorokhod, Oleksii A; Caione, Luisa; Migliardi, Giorgia; Barrera, Valentina; Piacibello, Wanda; Schwarzer, Evelin; Arese, Paolo; Smallegange, Renate C; Schmied, Wolfgang H; van Roey, Karel J; Verhulst, Niels O; Spitzen, Jeroen; Mukabana, Wolfgang R; Takken, Willem; Marin-Menendez, Alejandro; Bell, Angus; Biagini, Giancarlo A; Hill, Alasdair; Mbekeani, Alison; Shone, Alison; Nixon, Gemma; Stocks, Paul; Gibbons, Peter; Amewu, Richard; Hong, David W; Barton, Victoria; Pidathala, Chandra; Chadwick, James; Le Pensee, Louise; Warman, Ashley; Sharma, Raman; Fisher, Nick; Berry, Neil G; O'Neill, Paul M; Ward, Steve A; Brooke, Basil D; Kaiser, Maria L; Koekemoer, Lizette L; Coetzee, Maureen; Hunt, Richard H; Burgess, Steven J; Xu-Kelly, Jane; Liebmann, Katherine; Gunsaru, Bornface; Morrill, Westin; Peyton, David H; Chitnis, Nakul; Hardy, Diggory; Gnaegi, Guillaume; Boutsika, Konstantina; Maire, Nicolas; Steketee, Richard; Schapira, Allan; Smith, Tom; Tang, Jianxia; Inoue, Megumi; Sunahara, Toshihiko; Kanda, Moe; Kaneko, Osamu; Culleton, Richard; van Brummlen, Tharina; Becker, John VW; Mancama, Dalu T; Hoppe, Heinrich; Crosnier, Cecile; Wanaguru, Madushi; McDade, Brian; Rayner, Julian; Wright, Gavin J; de Oliveira, Alaíde Braga; Dolabela, Maria Fâni; Póvoa, Marinete Marins; Santos, Cid Aimbiré M; de Pilla Varotti, Fernando; Afolabi, Bamgboye M; Dunkwu, Antonia; Oparah, A C; Filipe, Ermelindo M; Antunes, Lina; Tomás, Esmael F; Viegas, Edna; Bernardo, João; Silva, Fortunato R; Tripathi, Abhai; Rienhoff, Hugh; Sullivan, David; Udagama-Randeniya, Preethi; Dias, Sajani; Premaratne, Prasad; Wickramarachchi, Thilan; Waitumbi, John; Nyakoe, Nancy; Muringo, Linda; Mahat, Ismail; Otiende, Moses; Susanna, Dewi; Eryando, Tris; Temidayo, Soniran O; Olufunmilayo, Idowu; Babatunde, Idowu A; Olusegun, Ajana; Tomás, Esmael; Filipe, E; Viegas, E; Sá, A; Silva, F; Antunes, L; Lafuente, E; Tonwong, Natda; Sattabongkot, Jetsumon; Sirichaisinthop, Jeeraphat; Udomsangpetch, Rachanee; Spjeldnæs, Astrid; Blomberg, Bjørn; Ginsburg, Hagai; Inoue, Megumi; Tang, Jianxia; Kaneko, Osamu; Yui, Katsuyuki; Culleton, Richard; Aubouy, Agnès; Kheliouen, Nabila; Tuikue-Ndam, Nicaise; Viwami, Firmine; Lalya, Francis; Eboumbou Moukoko, Else C; Rogier, Christophe; Deloron, Philippe; Omoregie, Ehimwenma S; Pal, Anirban; Darokar, Mahendra P; Chanda, Debabrata; Sisodia, Brijesh; Mogendi, Shem Oroo; Osman, Mamoun MM; Nour, Bakri YM; Sedig, Mohamed F; de Bes, Laura; Babikir, Adil M; Mohamedani, Ahmed A; Mens, Petra F; Ouédraogo, Alphonse; Coulibaly, Sheick O; Diarra, Amidou; Traoré, Abdoulaye; Sirima, Sodiomon B; Magnussen, Pascal; Ball, Elizabeth; Gonçalves, Carlos Penha; Pooe, Ofentse J; Shonhai, Addmore; Mharakurwa, Sungano; Roobsoong, Wanlapa; Roytrakul, Sittiruk; Kiatfuengfoo, Rachada; Nuchpramool, Wilairat; Cui, Liwang; Udomsangpetch, Rachanee; Schneider, Petra; Bell, Andy S; Read, Andrew F; Reece, Sarah E; Singh, Gavendra; Prakash, Soam; Siri, José G; Brown, Zachary; Spielauer, Martin; Rajasekariah, G-Halli R; Dogcio, Diane; Lee, Rogan; Hudson, Bernard J; Mazure, Hubert G; Smithyman, Anthony M; Rankin, Kathleen E; Tavares, Joana; Struck, Nicole S; Menard, Robert; Heussler, Volker T; Amino, Rogerio; Riglar, David; Richard, Dave; Boyle, Michelle; Wilson, Danny; Angrisano, Fiona; Turnbull, Lynne; Whitchurch, Cynthia; Cowman, Alan; Beeson, James; Ralph, Stuart; Baum, Jake; Rodrigues, Louise A; Henriques, Gisela; Cravo, Pedro; Prato, Mauro; Ulliers, Daniela; Gallo, Valentina; Schwarzer, Evelin; Akide-Ndunge, Oscar B; Mandili, Giorgia; Khadjavi, Amina; Saviozzi, Silvia; Calogero, Raffaele A; Arese, Paolo; Giribaldi, Giuliana; Bansal, Devendra; Herbert, Fabien; Deshpande, Prakash; Bécavin, Christophe; Guiyedi, Vincent; de Maria, Ilaria; Cazenave, Pierre-André; Mishra, Gyan Chandra; Ferlini, Cristiano; Fesel, Constantin; Benecke, Arndt; Pied, Sylviane; Hamid, Muzamil Mahdi Abdel; Remarque, Edmond J; Faber, Bart W; van Duivenvoorde, Leonie M; Kocken, Clemens HM; Thomas, Alan W; Houzé, Sandrine; Hubert, Véronique; Cohen, Pressler D; Rivetz, Baruch; Le Bras, Jacques; Jones, Matthew L; Collins, Mark O; Choudhary, Jyoti S; Rayner, Julian C; Koekemoer, Lizette L; Spillings, Belinda S; Christian, Riann; Wood, Oliver S; Kaiser, Maria; Norton, Ryan; Choi, Kwang S; Brooke, Basil D; Hunt, Richard H; Coetzee, Maureen; Gitau, Grace; Shonhai, Addmore; Dean Goldring, J P; Hurdayal, Ramona; Choveaux, David; Liehl, Peter; Prudêncio, Miguel; Carret, Céline; Mota, Maria M; Akter, Jasmin; Ahmed, Sabeena; Prue, Chai; Khan, Wasif; Sack, David; Haque, Rashidul; Sullivan, David; Kabanywany, Abdunoor Mulokozi; Mulure, Nathan; Migoha, Christopher; Malila, Aggrey; Lengeler, Christian; Schlienger, Raymond; Genton, Blaise; Niemand, J; Birkholtz, L; Louw, A I; Kirk, K; Ogonda, Lilian A; Orago, Alloys SS; Otieno, Michael F; Adhiambo, Christine; Otieno, Walter; Stoute, José A; Sutherland, Colin J; Oguike, Mary C; Smith, Valerie; Betson, Martha; Bousema, Teun; Chiodini, Peter L; Wells, Timothy NC; Takken, Willem; Cox-Singh, Janet; Crabb, Brendan; Bullen, Hayley; Charnaud, Sarah; Haase, Silvia; Boddey, Justin; Cowman, Alan; de Koning-Ward, Tania; Gilson, Paul; Tanner, Marcel; Alonso, Pedro L; van den Berg, Henk; Takken, Willem; Van den Steen, Philippe E; Geurts, Nathalie; Deroost, Katrien; Van Aelst, Ilse; Verhenne, Sebastien; Heremans, Hubertine; Van Damme, Jo; Opdenakker, Ghislain; Ward, Steve A; Fisher, Nicholas; Hill, Alasdair; Mbekeani, Alison; Shone, Alison; Nixon, Gemma; Stocks, Paul; Gibbons, Peter; Amewu, Richard; Hong, David W; Barton, Victoria; Pidathala, Chandra; Chadwick, James; Le Pensee, Louise; Warman, Ashley; Sharma, Raman; Berry, Neil G; O'Neill, Paul M; Biagini, Giancarlo A; Oyeyemi, Adebusola O; Alawode, Abdul-Gafar; Sogunro, Remi; Panichakul, Tasanee; Payuhakrit, Witchuda; Wongborisuth, Chokdee; Hongeng, Suradej; Udomsangpetch, Rachanee; Parikh, Ravi; Amole, Isaac; Tarpley, Margaret; Gbadero, Daniel; Davidson, Mario; Vermund, Sten H; Patzewitz, Eva-Maria; Müller, Sylke; Noor, Ramadhani A; Thiesen, Michael; Mordmuller, Benjamin; Milligan, Paul; Atuguba, Frank; Sirima, Sodiomon; Issifou, Saadou; Bojang, Kalifa; Kironde, Fred; Tiono, Alfred; Okech, Brenda; Chilengi, Roma; Ngoa, Ateba; Mukasa, Kaddu; Jepsen, Soren; Ochola, Lucy B; Siddondo, Bethsheba R; Ocholla, Harold; Nyka, Siana; Kimani, Eva N; Williams, Thomas N; Makale, Johnstone O; Liljander, Anne; Urban, Britta C; Bull, Pete; Szestak, Tadge; Marsh, Kevin; Craig, Alister G; Malisa, Allen; Pearce, Richard; Abdullah, Salim; Mshinda, Hassan; Kachur, Patrick; Bloland, Peter; Roper, Cally; Mbugi, Erasto V; Meijerink, Marjolein; Veenemans, Jacobien; Jeurink, Prescilla V; McCall, Matthew; Olomi, Raimos M; Shao, John F; Chilongola, Jaffu O; Verhoef, Hans; Savelkoul, Huub FJ; Mirghani, Samia E; Nour, Bakri YM; Bushra, Sayed M; Hassan, Ibrahim El; Snow, Robert W; Noor, Abdisalan M; Mnyone, Ladslaus L; Lyimo, Issa N; Lwetoijera, Dickson W; Mpingwa, Monica W; Nchimbi, Nuru; Hancock, Penny; Russell, Tanya L; Kirby, Matthew J; Takken, Willem; Koenraadt, Constantianus JM; Odhiambo, Collins O; Otieno, Walter; Adhiambo, Christine; Odera, Michael M; Stoute, José A; Ferrer, Jordi; Prats, Clara; López, Daniel; Valls, Joaquim; Gargallo, Domingo; Wijayalath, Wathsala; Cheesman, Sandie; Rajakaruna, Jagath; Weerasinghe, Sudath; Kapilananda, Gamini; Gamage, Kamal; Perera, Kamal; Handunnetti, Shiroma; Carter, Richard; Pathirana, Sisira; Wanjala, Christine L; Githeko, Andrew K; Waitumbi, John N; Gomes-Santos, Carina SS; Braks, J Anneke M; Prudêncio, Miguel; Carret, Céline K; Gomes, Ana Rita; Pain, Arnab; Feltwell, Theresa; Khan, Shahid M; Waters, Andrew P; Janse, Chris J; Mair, Gunnar R; Mota, Maria M; Kyabayinze, Daniel J; Asiimwe, Caroline; Nakanjako, Damalie; Nabakooza, Jane; Counihan, Helen; Tibenderana, James K; Donegan, G; Forrester, C A; Ward, S A; Boyom, Fabrice F; Madiesse, Eugénie K; Bankeu, Jean J; Tsouh, Valere P; Lenta, Bruno N; Mbacham, Wilfred F; Tsamo, Etienne; Zollo, Paul HA; Gut, Jiri; Rosenthal, Philip J; Yoon, Ho Sup; Alag, Reema; Kang, Congbao; Ye, Hong; Kotaka, Masayo; Qureshi, Insaf A; Bharatham, Nagakumar; Shin, Joon; Bozdech, Zbynek; Preiser, Peter; Lescar, Julien; Wanaguru, Madushi; Wright-Crosnier, Cecile; Bustamante, Leyla; McDade, Brian; Rayner, Julian; Wright, Gavin J; Crowell, Valerie; Hardy, Diggory; Chitnis, Nakul; Maire, Nicolas; Smith, Thomas