日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A yeast two-hybrid system for the screening and characterization of small-molecule inhibitors of protein-protein interactions identifies a novel putative Mdm2-binding site in p53

用于筛选和表征蛋白质-蛋白质相互作用的小分子抑制剂的酵母双杂交系统鉴定了 p53 中一个新的假定的 Mdm2 结合位点

Jin Huei Wong, Mohammad Alfatah, Mei Fang Sin, Hong May Sim, Chandra S Verma, David P Lane, Prakash Arumugam

ARRY-334543 reverses multidrug resistance by antagonizing the activity of ATP-binding cassette subfamily G member 2

ARRY-334543 通过拮抗 ATP 结合盒亚家族 G 成员 2 的活性来逆转多药耐药性

De-Shen Wang, Atish Patel, Hong-May Sim, Yun-Kai Zhang, Yi-Jun Wang, Rishil J Kathawala, Hui Zhang, Tanaji T Talele, Suresh V Ambudkar, Rui-Hua Xu, Zhe-Sheng Chen

Saracatinib (AZD0530) is a potent modulator of ABCB1-mediated multidrug resistance in vitro and in vivo

Saracatinib (AZD0530) 是体外和体内 ABCB1 介导的多药耐药性的强效调节剂

Ke-Jun Liu, Jie-Hua He, Xiao-Dong Su, Hong-May Sim, Jing-Dun Xie, Xing-Gui Chen, Fang Wang, Yong-Ju Liang, Satyakam Singh, Kamlesh Sodani, Tanaji T Talele, Suresh V Ambudkar, Zhe-Sheng Chen, Hai-Ying Wu, Li-Wu Fu