Discovery of a novel Na(v)1.5 inhibitor reducing cardiac conduction via structure-based virtual screening and assays
通过基于结构的虚拟筛选和检测,发现了一种新型的Na(v)1.5抑制剂,该抑制剂可降低心脏传导。
期刊:Acta Pharmacologica Sinica
影响因子:8.4
doi:10.1038/s41401-025-01679-4
Wang, Ying-Ying; Wang, Gao-Ang; You, Qing; Liu, Yi-Fei; Qu, Wang-Lin; Chen, Yi-Hong; Mu, Chen-Zhang; Zhou, Xi; Liu, Min; Yang, Wei; Hou, Ting-Jun