Identification of a Novel Linker Enabling the Bioconjugation of a Cyclic Dinucleotide for the STING Antibody-Drug Conjugate TAK-500
鉴定一种新型连接子,用于STING抗体-药物偶联物TAK-500的环状二核苷酸生物偶联
期刊:Bioconjugate Chemistry
影响因子:3.9
doi:10.1021/acs.bioconjchem.5c00424
Lee, Hong Myung; Abdul-Hadi, Kojo; Appleman, Vicky A; Cardin, David; Dong, Linlin; England, Dylan; Ganno, Michelle L; Gershman, Rachel; Gigstad, Kenneth; Gulavita, Nanda; Hu, Zhigen; Huang, Jian; Huang, Shih-Chung; Lok, David; Ma, Liting; Malley, Jenna; Mizutani, Miho; Molchanova, Nina; Piatkov, Konstantin I; Rice, Elise; Shi, Zhan; Vyskocil, Stepan; Wang, Jianing; Xu, He; Xu, Tianlin; Zhang, Dong Mei; Zhang, Ji; Abu-Yousif, Adnan O