日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cellular Target Engagement and Dissociation Kinetics of Class I-Selective Histone Deacetylase (HDAC) Inhibitors

I类选择性组蛋白去乙酰化酶(HDAC)抑制剂的细胞靶点结合和解离动力学

Honin, Irina; Novakova, Zora; Feller, Felix; Schneider, Simon; Schäker-Hübner, Linda; Barinka, Cyril; K Hansen, Finn

Development of the First-in-Class FEM1B-Recruiting Histone Deacetylase Degraders

首创的FEM1B募集组蛋白去乙酰化酶降解剂的开发

Felix Feller ,Irina Honin ,Martina Miranda ,Heiko Weber ,Svenja Henze ,Maria Hanl ,Finn K Hansen

Development and Characterization of the First Selective Class IIb Histone Deacetylase Degraders.

首个选择性 IIb 类组蛋白去乙酰化酶降解剂的开发和表征

Zhai Shiyang, Honin Irina, Schäker-Hübner Linda, Hanl Maria, Jacobi Lukas, Dressler Finn, Pieńkowska Dominika Ewa, König Philipp, Gerhartz Jan, Voget Rabea, Bendas Gerd, Gütschow Michael, Meissner Felix, Burckhardt Bjoern B, Nowak Radosław P, Steinebach Christian, Hansen Finn K

Targeted Degradation of Histone Deacetylases via Bypassing E3 Ligase Targeting Chimeras (BYETACs)

通过绕过 E3 连接酶靶向嵌合体 (BYETACs) 靶向降解组蛋白去乙酰化酶

Sun, Tao; Zhai, Shiyang; König, Beate; Honin, Irina; Kponomaizoun, Cindy-Esther; Hansen, Finn K

Development of Ethyl-Hydrazide-Based Selective Histone Deacetylase 6 (HDAC6) PROTACs

基于乙肼的选择性组蛋白去乙酰化酶6 (HDAC6) PROTACs 的开发

Stopper, Daniel; Honin, Irina; Feller, Felix; Hansen, Finn K

Target Engagement Studies and Kinetic Live-Cell Degradation Assays Enable the Systematic Characterization of Histone Deacetylase 6 Degraders

靶标结合研究和动力学活细胞降解分析能够系统地表征组蛋白去乙酰化酶 6 降解剂

Hanl, Maria; Feller, Felix; Honin, Irina; Tan, Kathrin; Miranda, Martina; Schäker-Hübner, Linda; Bückreiß, Nico; Schiedel, Matthias; Gütschow, Michael; Bendas, Gerd; Hansen, Finn K

Ortho-Hydroxyanilides: Slow-Acting, Selective Histone Deacetylase 1/2 Inhibitors Suitable for Photocaging Applications

邻羟基苯胺类化合物:作用缓慢、选择性的组蛋白去乙酰化酶1/2抑制剂,适用于光笼应用

Honin, Irina; Sun, Tao; Setia, Nisha; Schäker-Hübner, Linda; Hansen, Finn K

DCAF16-Based Covalent Molecular Glues for Targeted Protein Degradation of Histone Deacetylases.

基于DCAF16的共价分子胶用于靶向降解组蛋白去乙酰化酶

Sun Tao, Zhai Shiyang, Lepper Stephan, König Beate, Malenica Mateo, Honin Irina, Hansen Finn K

Replacing a Cereblon Ligand by a DDB1 and CUL4 Associated Factor 11 (DCAF11) Recruiter Converts a Selective Histone Deacetylase 6 PROTAC into a Pan-Degrader

用 DDB1 和 CUL4 相关因子 11 (DCAF11) 募集因子取代 Cereblon 配体,可将选择性组蛋白去乙酰化酶 6 PROTAC 转化为泛降解酶。

Feller, Felix; Weber, Heiko; Miranda, Martina; Honin, Irina; Hanl, Maria; Hansen, Finn K

Impact of Distal Protection with Filter-Type Device on Long-term Outcome after Percutaneous Coronary Intervention for Acute Myocardial Infarction: Clinical Results with Filtrap®

采用滤器型装置进行远端保护对急性心肌梗死经皮冠状动脉介入治疗后长期预后的影响:Filtrap® 的临床结果

Ryota Teramoto,Kenji Sakata, Kenji Miwa, Takao Matsubara, Toshihiko Yasuda, Masaru Inoue, Hirofumi Okada, Honin Kanaya, Masa-Aki Kawashiri, Masakazu Yamagishi, Kenshi Hayashi