日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of BI-2493, a Pan-KRAS Inhibitor Showing In Vivo Efficacy.

发现 BI-2493,一种泛 KRAS 抑制剂,显示出体内疗效

Bröker Joachim, Waterson Alex G, Hodges Timothy R, Abbott Jason R, Arnold Allison, Böttcher Jark, Braun Nina, Cui Jianwen, Fuchs Julian E, Gerstberger Thomas, Gogg Sebastian, Hanner Sabine, Herdeis Lorenz, Howell Lucas W, Mantoulidis Andreas, Mayer Moriz, Phan Jason, Rocchetti Francesca, Sankar Kyra, Sarkar Dhruba, Schaaf Otmar, Sensintaffar John L, Sun Qi, Wunberg Tobias, Fesik Stephen W

Stereospecific access to α-haloalkyl esters via enol ester epoxides and synthesis of a C3-C21 fragment of bastimolide A

通过烯醇酯环氧化物立体选择性合成α-卤代烷基酯,并合成巴斯蒂莫利德A的C3-C21片段

Howell, Lucas W; Hackbarth, Jacob N; Abraham, Jeffrey S; Friestad, Gregory K