日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification and Biological Evaluation of a Novel CLK4 Inhibitor Targeting Alternative Splicing in Pancreatic Cancer Using Structure-Based Virtual Screening.

利用基于结构的虚拟筛选方法鉴定和生物学评价一种靶向胰腺癌中选择性剪接的新型 CLK4 抑制剂

Yang Chun-Lin, Wu Yi-Wen, Tu Huang-Ju, Yeh Yun-Hsuan, Lin Tony Eight, Sung Tzu-Ying, Li Mu-Chun, Yen Shih-Chung, Hsieh Jui-Hua, Yu Ming-Chin, Hsieh Sen-Yung, Hsieh Hsing-Pang, Pan Shiow-Lin, Hsu Kai-Cheng

Noncovalent Interaction Effects on the Acyl Radical Reaction of Bicyclo[2.2.2]octanone: Selective Formation of Rearrangement and Cyclization Products

非共价相互作用对双环[2.2.2]辛酮酰基自由基反应的影响:重排和环化产物的选择性生成

Chen, Chih-Ming; Kuo, Tung-Chun; Reddy, Julakanti Satyanarayana; Teoh, Yi Ning; Huang, Jyun-Sian; Lin, Sheng-Kuo; Cheng, Mu-Jeng; Hsieh, Hsing-Pang

Integrating machine learning and protein-ligand interaction profiling for the discovery of METTL3 inhibitors

整合机器学习和蛋白质-配体相互作用分析以发现METTL3抑制剂

Huang, Wei-Cheng; Hsieh, Hsing-Pang; Tung, Chun-Wei

Influence of Ring Strain on the Formation of Rearrangement vs Cyclization Isotwistane Products in the Acyl Radical Reaction of Bicyclo[2.2.2]octanone

环张力对双环[2.2.2]辛酮酰基自由基反应中重排与环化异扭烷产物形成的影响

Chen, Chih-Ming; Lin, Sheng-Kuo; Hsieh, Chi-Tien; Reddy, Julakanti Satyanarayana; Teoh, Yi Ning; Cheng, Mu-Jeng; Hsieh, Hsing-Pang

A critical overview of current progress for COVID-19: development of vaccines, antiviral drugs, and therapeutic antibodies

对当前新冠肺炎研究进展的关键概述:疫苗、抗病毒药物和治疗性抗体的研发

Kumari, Monika; Lu, Ruei-Min; Li, Mu-Chun; Huang, Jhih-Liang; Hsu, Fu-Fei; Ko, Shih-Han; Ke, Feng-Yi; Su, Shih-Chieh; Liang, Kang-Hao; Yuan, Joyce Pei-Yi; Chiang, Hsiao-Ling; Sun, Cheng-Pu; Lee, I-Jung; Li, Wen-Shan; Hsieh, Hsing-Pang; Tao, Mi-Hua; Wu, Han-Chung

Briarenols W-Z: Chlorine-Containing Polyoxygenated Briaranes from Octocoral Briareum stechei (Kükenthal, 1908)

Briarenols WZ:来自八放珊瑚 Briareum stechei (Kükenthal, 1908) 的含氯多氧 Briaranes

Chen, You-Ying; Zhang, Yi-Lin; Lee, Gene-Hsiang; Tsou, Lun Kelvin; Zhang, Mingzi M; Hsieh, Hsing-Pang; Chen, Jih-Jung; Ko, Chou-Yuan; Wen, Zhi-Hong; Sung, Ping-Jyun

Mimicking H3 Substrate Arginine in the Design of G9a Lysine Methyltransferase Inhibitors for Cancer Therapy: A Computational Study for Structure-Based Drug Design

在癌症治疗中,通过模拟H3底物精氨酸来设计G9a赖氨酸甲基转移酶抑制剂:基于结构的药物设计的计算研究

Chandar Charles, M Ramya; Li, Mu-Chun; Hsieh, Hsing-Pang; Coumar, Mohane Selvaraj

Design of drug-like hepsin inhibitors against prostate cancer and kidney stones

设计用于治疗前列腺癌和肾结石的类药物肝素抑制剂

Blay, Vincent; Li, Mu-Chun; Ho, Sunita P; Stoller, Mashall L; Hsieh, Hsing-Pang; Houston, Douglas R

Targeting P-glycoprotein: Investigation of piperine analogs for overcoming drug resistance in cancer

靶向P-糖蛋白:胡椒碱类似物在克服癌症耐药性方面的研究

Syed, Safiulla Basha; Arya, Hemant; Fu, I-Hsuan; Yeh, Teng-Kuang; Periyasamy, Latha; Hsieh, Hsing-Pang; Coumar, Mohane Selvaraj

Homology modeling of DFG-in FMS-like tyrosine kinase 3 (FLT3) and structure-based virtual screening for inhibitor identification

DFG-in FMS样酪氨酸激酶3 (FLT3) 的同源建模及基于结构的抑制剂筛选

Ke, Yi-Yu; Singh, Vivek Kumar; Coumar, Mohane Selvaraj; Hsu, Yung Chang; Wang, Wen-Chieh; Song, Jen-Shin; Chen, Chun-Hwa; Lin, Wen-Hsing; Wu, Szu-Huei; Hsu, John T A; Shih, Chuan; Hsieh, Hsing-Pang