日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A small molecule VDAC ligand inhibits ERAD and induces selective cancer cell death via disruption of calcium homeostasis.

一种小分子 VDAC 配体通过破坏钙稳态抑制 ERAD 并诱导选择性癌细胞死亡。

Yan Wenjing, Talley Daniel C, Syam Antara, Danchik Carina, Zhong Yongwang, Zhang Xianzheng, Liu Xiaoying, Baljinnyam Bolormaa, Kales Stephen C, Cyr Matthew G, Fang Yuhong, Zakharov Alexey V, Hu Xin, Niehoff Taylor, Xu Tuan, Qu Yanyan, Yang Allison, Courouble Valentine V, Yao Qin, Simeonov Anton, Huang Ruili, Rostovtseva Tatiana K, Bezrukov Sergey M, LeClair Christopher A, Egan Josephine M, Wang Hua, Tao Dingyin, Rai Ganesha, Henderson Mark J, Fang Shengyun

Quantitative high-throughput screening identifies small-molecule modulators of Wnt/β-catenin signaling

定量高通量筛选鉴定Wnt/β-catenin信号通路的小分子调节剂

Chen, Xing; Yang, Shu; Sakamuru, Srilatha; Sukhawanit, Chainarong; Wood, Savannah; Ooka, Masato; Huang, Ruili; Xia, Menghang

Identifying androgen receptor antagonists using a metabolically competent high-throughput screening assay

利用代谢能力强的高通量筛选方法鉴定雄激素受体拮抗剂

Lynch, Caitlin; Shah, Pranav; Zhao, Jinghua; Xu, Xin; Huang, Ruili; Xia, Menghang

Profiling of Environmental Mixtures Containing Metals for Their Toxicity Pathways and Mechanism of Action

对含金属环境混合物的毒性途径和作用机制进行分析

Ooka, Masato; Zhao, Jinghua; Zhang, Li; Huang, Ruili; Sakamuru, Srilatha; TeKrony, Charlotte; Hsieh, Jui-Hua; Collins, Bradley J; Dunnick, June K; Dixon, Darlene; Xia, Menghang

Expanded Tox21 biological assay panel for the prediction of drug-induced liver injury and cardiotoxicity

用于预测药物性肝损伤和心脏毒性的扩展型 Tox21 生物检测组合

Xu, Tuan; Ooka, Masato; Zhao, Jinghua; Sakamuru, Srilatha; Ngan, Deborah K; Zhang, Li; Yang, Shu; Travers, Jameson; Xia, Menghang; Zhao, Tongan; Klumpp-Thomas, Carleen; Zhu, Hu; Hall, Mathew D; Ferguson, Stephen; Shaw, Natalie D; Reif, David M; Simeonov, Anton; Huang, Ruili

Leveraging viral genome sequences and machine learning models for identification of potentially selective antiviral agents

利用病毒基因组序列和机器学习模型来识别潜在的选择性抗病毒药物

Xu, Tuan; Xu, Miao; Zhang, Qi; Chen, Catherine Z; Zheng, Wei; Huang, Ruili

Genetic Variants of GBP4: Reduced Risks for Drug-Induced Acute Liver Failure in Non-Finnish European Population

GBP4基因变异:降低非芬兰裔欧洲人群药物诱发急性肝衰竭的风险

Liao, Tsung-Jen; Xia, Menghang; Hayashi, Paul; Pan, Bohun; Aithal, Guruprasad P; Lucena, M Isabel; Andrade, Raúl J; Rule, Jody A; Lee, William M; Rakela, Jorge; Huang, Ruili; Chen, Minjun

The threshold effect of fasting blood glucose levels on the risk of delivering macrosomia in gestational diabetes mellitus patients

空腹血糖水平阈值效应对妊娠期糖尿病患者分娩巨大儿风险的影响

Li, Yuan; Zhu, Yumin; Zheng, Wenjun; Gao, Yumei; Huang, Ruili; Yang, Tingting; Chen, Ying

Lessons learned from evaluating defined chemical mixtures in a high-throughput estrogen receptor assay system

从高通量雌激素受体检测系统中评估特定化学混合物所汲取的经验教训

Parham, Fred; Eccles, Kristin M; Rider, Cynthia V; Sakamuru, Srilatha; Xia, Menghang; Huang, Ruili; Tice, Raymond R; Dinse, Gregg E; DeVito, Michael J

ICRF193 potentiates the genotoxicity of etoposide

ICRF193 可增强依托泊苷的遗传毒性

Ooka, Masato; Mitchell, Leah; Zhao, Jinghua; Hirota, Kouji; Huang, Ruili; Abe, Takuya; Xia, Menghang