Tetrafluorophenoxymethyl ketone cruzain inhibitors with improved pharmacokinetic properties as therapeutic leads for Chagas' disease
具有改善的药代动力学特性的四氟苯氧甲基酮类克鲁兹蛋白酶抑制剂可作为治疗恰加斯病的先导化合物
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2015.06.066
Neitz, R Jeffrey; Bryant, Clifford; Chen, Steven; Gut, Jiri; Hugo Caselli, Estefania; Ponce, Servando; Chowdhury, Somenath; Xu, Haichao; Arkin, Michelle R; Ellman, Jonathan A; Renslo, Adam R