日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Slow conformational dynamics of the human A2A adenosine receptor are temporally ordered

人类A2A腺苷受体的缓慢构象动力学具有时间有序性。

Shushu Wei ,Naveen Thakur ,Arka P Ray ,Beining Jin ,Samuel Obeng ,Christopher R McCurdy ,Lance R McMahon ,Hugo Gutiérrez-de-Terán ,Matthew T Eddy ,Rajan Lamichhane

Potent and Subtype-Selective Dopamine D2 Receptor Biased Partial Agonists Discovered via an Ugi-Based Approach

通过基于 Ugi 的方法发现强效且亚型选择性的多巴胺 D2 受体偏向部分激动剂

Ana Mallo-Abreu, Irene Reyes-Resina, Jhonny Azuaje, Rafael Franco, Aitor García-Rey, Maria Majellaro, Darío Miranda-Pastoriza, Xerardo García-Mera, Willem Jespers, Hugo Gutiérrez-de-Terán, Gemma Navarro, Eddy Sotelo

Design, synthesis, HER2 inhibition and anticancer evaluation of new substituted 1,5-dihydro-4,1-benzoxazepines

新型取代 1,5-二氢-4,1-苯并氧氮卓类药物的设计、合成、HER2 抑制及抗癌评价

Olga Cruz-López, Matilde Ner, Francho Nerín-Fonz, Yaiza Jiménez-Martínez, David Araripe, Juan A Marchal, Houria Boulaiz, Hugo Gutiérrez-de-Terán, Joaquín M Campos, Ana Conejo-García

Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors

取代螺环吲哚二氢喹唑啉酮作为 IRAP 抑制剂的合成、评价及建议结合位点

Karin Engen, Sudarsana Reddy Vanga, Thomas Lundbäck, Faith Agalo, Vivek Konda, Annika Jenmalm Jensen, Johan Åqvist, Hugo Gutiérrez-de-Terán, Mathias Hallberg, Mats Larhed, Ulrika Rosenström

The GPR139 reference agonists 1a and 7c, and tryptophan and phenylalanine share a common binding site

GPR139 参考激动剂 1a 和 7c,以及色氨酸和苯丙氨酸共享一个共同的结合位点

Anne Cathrine Nøhr, Willem Jespers, Mohamed A Shehata, Leonard Floryan, Vignir Isberg, Kirsten Bayer Andersen, Johan Åqvist, Hugo Gutiérrez-de-Terán, Hans Bräuner-Osborne, David E Gloriam

Recombinant plasmepsin 1 from the human malaria parasite plasmodium falciparum: enzymatic characterization, active site inhibitor design, and structural analysis

来自人类疟原虫恶性疟原虫的重组疟原虫蛋白酶 1:酶学特性、活性位点抑制剂设计和结构分析

Peng Liu, Melissa R Marzahn, Arthur H Robbins, Hugo Gutiérrez-de-Terán, David Rodríguez, Scott H McClung, Stanley M Stevens Jr, Charles A Yowell, John B Dame, Robert McKenna, Ben M Dunn