Using the Scaffold of FDA-Approved Drugs with Trypanocidal Activity to Identify New Anti-Trypanosoma cruzi Agents: An In Silico and In Vitro Approach
利用已获FDA批准的具有锥虫杀灭活性的药物骨架来鉴定新的抗克氏锥虫药物:一种计算机模拟和体外方法
期刊:Cell
影响因子:42.5
doi:10.1016/j.cell.2026.02.017
Yamamuro, Tadashi; Katoh, Daisuke; Silva, Guilherme Martins; Nishida, Hiroshi; Oikawa, Satoshi; Higuchi, Yusuke; Wang, Dandan; Fujimoto, Masanori; Yoshida, Naofumi; Li, Mark; Shin, Jihoon; Zhao, Zezhou; Yook, Jin-Seon; Sun, Lijun; Kajimura, Shingo; Xie, Qingchao; Liu, Yihui; Zhang, Zhe; Zhang, Hongmin; Xu, Jin; Wang, Yeru; Zhao, Yong; Zhao, Qingxia; Song, Jingyi; Li, Xukai; Zhang, Zhongwei; Xiao, Junsong; Wu, Hua; Huang, Mingquan; Boppana, Sri Harsha; Luke, Naveena; Karuchola, Sravani; Udaikumar, Jahnavi; Mintz, Cyrus David; Zhou, Yaxi; Xu, Dong; Bu, Meichao; Li, Ke; Gao, Lingyu; Pan, Fei; Peng, Wenjun; Chen, Hualei; Tian, Wenli; Lyu, Yipin; Zhang, Jie; Cheng, Chi; Tang, Xue; Huang, Pantian; Liu, Feitong; Hu, Ruibiao; Huppertz, Thom; Wang, Xinyan; Zhou, Peng; Zhang, Xiaojing; Xing, Huizhen; Liu, Huiping; Zhang, Xiaowei; Vázquez-Jiménez, Lenci K; González-González, Alonzo; Delgado-Maldonado, Timoteo; Gómez-Escobedo, Rogelio; Avalos-Navarro, Guadalupe; Moreno-Rodríguez, Adriana; Paz-González, Alma D; Ortiz-Pérez, Eyra; Nogueda-Torres, Benjamín; Rivera, Gildardo