日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

3'-deoxytubercidin: A potent therapeutic candidate for the treatment of Surra and Dourine

3'-脱氧结核菌素:一种治疗苏拉病和杜林病的有效候选药物

Ilbeigi, Kayhan; Mabille, Dorien; Roy, Rajdeep; Bundschuh, Mirco; Van de Velde, Ewout; Hulpia, Fabian; Van Calenbergh, Serge; Caljon, Guy

Ex Vivo Feedback Control of Neurotransmission Using a Photocaged Adenosine A1 Receptor Agonist

利用光笼腺苷A1受体激动剂进行离体神经传递反馈控制

Craey, Erine; Hulpia, Fabian; Spanoghe, Jeroen; Manzella, Simona; Larsen, Lars E; Sprengers, Mathieu; De Bundel, Dimitri; Smolders, Ilse; Carrette, Evelien; Delbeke, Jean; Vonck, Kristl; Boon, Paul; Van Calenbergh, Serge; Wadman, Wytse J; Raedt, Robrecht

4E Interacting Protein as a Potential Novel Drug Target for Nucleoside Analogues in Trypanosoma brucei

4E 相互作用蛋白作为布氏锥虫核苷类似物的潜在新型药物靶点

Dorien Mabille, Camila Cardoso Santos, Rik Hendrickx, Mathieu Claes, Peter Takac, Christine Clayton, Sarah Hendrickx, Fabian Hulpia, Louis Maes, Serge Van Calenbergh, Guy Caljon

7-Aryl-7-deazapurine 3'-deoxyribonucleoside derivative as a novel lead for Chagas' disease therapy: in vitro and in vivo pharmacology

7-芳基-7-脱氮嘌呤3'-脱氧核糖核苷衍生物作为治疗恰加斯病的新型先导化合物:体外和体内药理学研究

Cardoso-Santos, Camila; Ferreira de Almeida Fiuza, Ludmila; França da Silva, Cristiane; Mazzeti, Ana Lia; Donola Girão, Roberson; Melo de Oliveira, Gabriel; da Gama Jaen Batista, Denise; Cruz Moreira, Otacilio; Lins da Silva Gomes, Natália; Maes, Louis; Caljon, Guy; Hulpia, Fabian; Calenbergh, Serge V; Correia Soeiro, Maria de Nazaré

Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents

将结核分枝杆菌胸苷酸激酶 (MtbTMPK) 抑制剂转化为潜在抗分枝杆菌药物的努力

Jian, Yanlin; Merceron, Romain; De Munck, Steven; Forbes, He Eun; Hulpia, Fabian; Risseeuw, Martijn D P; Van Hecke, Kristof; Savvides, Savvas N; Munier-Lehmann, Hélène; Boshoff, Helena I M; Van Calenbergh, Serge

New fluoroethyl phenylalanine analogues as potential LAT1-targeting PET tracers for glioblastoma

新型氟乙基苯丙氨酸类似物可作为胶质母细胞瘤的潜在 LAT1 靶向 PET 示踪剂

Jeroen Verhoeven, Fabian Hulpia, Ken Kersemans, Julie Bolcaen, Stef De Lombaerde, Jan Goeman, Benedicte Descamps, Giorgio Hallaert, Caroline Van den Broecke, Karel Deblaere, Christian Vanhove, Johan Van der Eycken, Serge Van Calenbergh, Ingeborg Goethals, Filip De Vos

Synthesis of a 3'-C-ethynyl-β-d-ribofuranose purine nucleoside library: Discovery of C7-deazapurine analogs as potent antiproliferative nucleosides

3'-C-乙炔基-β-D-呋喃核糖嘌呤核苷库的合成:发现C7-脱氮嘌呤类似物作为强效抗增殖核苷

Hulpia, Fabian; Noppen, Sam; Schols, Dominique; Andrei, Graciela; Snoeck, Robert; Liekens, Sandra; Vervaeke, Peter; Van Calenbergh, Serge

Exploring the purine core of 3'-C-ethynyladenosine (EAdo) in search of novel nucleoside therapeutics

探索3'-C-乙炔基腺苷(EAdo)的嘌呤核心结构,以寻找新型核苷类药物

Hulpia, Fabian; Balzarini, Jan; Schols, Dominique; Andrei, Graciela; Snoeck, Robert; Van Calenbergh, Serge