日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

Perspectives of the Obstetric Care Environment for Pregnant Individuals Who Have an Opioid Use Disorder

对患有阿片类药物使用障碍的孕妇的产科护理环境的看法

Girasulo, Samantha; Maltz, Caro; Weichert, Maggie; Kaufman, Joy S; Mele, Amanda; Hunkele, Karen; Yonkers, Kimberly A; Byatt, Nancy; Forray, Ariadna

Oxa-Iboga alkaloids lack cardiac risk and disrupt opioid use in animal models

Oxa-Iboga 生物碱在动物模型中不具有心脏风险,并能干扰阿片类药物的使用

Václav Havel #, Andrew C Kruegel #, Benjamin Bechand #, Scot McIntosh, Leia Stallings, Alana Hodges, Madalee G Wulf, Mel Nelson, Amanda Hunkele, Michael Ansonoff, John E Pintar, Christopher Hwu, Rohini S Ople, Najah Abi-Gerges, Saheem A Zaidi, Vsevolod Katritch, Mu Yang, Jonathan A Javitch, Susruta

Site selective C-H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy

帽柱木碱的位点选择性CH官能化揭示了一种调节阿片受体信号传导效力的分子开关

Bhowmik, Srijita; Galeta, Juraj; Havel, Václav; Nelson, Melissa; Faouzi, Abdelfattah; Bechand, Benjamin; Ansonoff, Mike; Fiala, Tomas; Hunkele, Amanda; Kruegel, Andrew C; Pintar, John E; Majumdar, Susruta; Javitch, Jonathan A; Sames, Dalibor

Oxidative Metabolism as a Modulator of Kratom's Biological Actions

氧化代谢作为 Kratom 生物作用的调节剂

Soumen Chakraborty, Rajendra Uprety, Samuel T Slocum, Takeshi Irie, Valerie Le Rouzic, Xiaohai Li, Lisa L Wilson, Brittany Scouller, Amy F Alder, Andrew C Kruegel, Michael Ansonoff, Andras Varadi, Shainnel O Eans, Amanda Hunkele, Abdullah Allaoa, Sanjay Kalra, Jin Xu, Ying Xian Pan, John Pintar, Bro

Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site

通过靶向正位点的不同亚区来控制阿片受体功能选择性

Rajendra Uprety #, Tao Che #, Saheem A Zaidi #, Steven G Grinnell, Balázs R Varga, Abdelfattah Faouzi, Samuel T Slocum, Abdullah Allaoa, András Varadi, Melissa Nelson, Sarah M Bernhard, Elizaveta Kulko, Valerie Le Rouzic, Shainnel O Eans, Chloe A Simons, Amanda Hunkele, Joan Subrath, Ying Xian Pan, 

Correction to: Mu Opioids Induce Biased Signaling at the Full-Length Seven Transmembrane C-Terminal Splice Variants of the mu Opioid Receptor Gene, Oprm1

更正:μ阿片受体在μ阿片受体基因Oprm1的全长七次跨膜C端剪接变体处诱导偏向性信号传导

Narayan, Ankita; Hunkele, Amanda; Xu, Jin; Bassoni, Daniel L; Pasternak, Gavril W; Pan, Ying-Xian

Kratom Alkaloids as Probes for Opioid Receptor Function: Pharmacological Characterization of Minor Indole and Oxindole Alkaloids from Kratom

卡痛叶生物碱作为阿片类受体功能探针:卡痛叶中次要吲哚和氧吲哚生物碱的药理学表征

Soumen Chakraborty, Rajendra Uprety, Amal E Daibani, Valerie L Rouzic, Amanda Hunkele, Kevin Appourchaux, Shainnel O Eans, Nitin Nuthikattu, Rahul Jilakara, Lisa Thammavong, Gavril W Pasternak, Ying-Xian Pan, Jay P McLaughlin, Tao Che, Susruta Majumdar

Mu Opioids Induce Biased Signaling at the Full-Length Seven Transmembrane C-Terminal Splice Variants of the mu Opioid Receptor Gene, Oprm1

Mu 阿片类药物在 mu 阿片类受体基因 Oprm1 的全长七个跨膜 C 末端剪接变体处诱导偏向信号传导

Ankita Narayan, Amanda Hunkele, Jin Xu, Daniel L Bassoni, Gavril W Pasternak, Ying-Xian Pan

Pharmacological characterization of novel synthetic opioids (NSO) found in the recreational drug marketplace

娱乐性药物市场上发现的新型合成阿片类药物 (NSO) 的药理学表征

Michael H Baumann, Susruta Majumdar, Valerie Le Rouzic, Amanda Hunkele, Rajendra Uprety, Xi Ping Huang, Jin Xu, Bryan L Roth, Ying-Xian Pan, Gavril W Pasternak