日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Pharmacology of a Morphinan-Derived Dual Mu-Kappa Opioid Receptor Agonist Analgesic.

吗啡烷衍生的双重μ-κ阿片受体激动剂镇痛药的合成与药理学研究

Varga Balazs R, Uprety Rajendra, Paul Barnali, Knoll Alexis, Ramos-Gonzalez Nokomis, Appourchaux Kevin, Taylor Tori, Turgutalp Bengisu, Shinouchi Ryosuke, Eans Shainnel O, Williams Ashai K, Vasquez-Grinnell Steven G, Zaidi Saheem, Nazarova Antonina L, Varadi Andras, Le Rouzic Valerie, Brown Taylor G, Martinez Shani, Ansonoff Michael, Dardashti Rebecca Notis, Hunkele Amanda, Subrath Joan, Welch Matthew, Xu Jin, Rossi Grace C, Pintar John, Pasternak Gavril W, Katritch Vsevolod, McLaughlin Jay P, Pan Ying Xian, Majumdar Susruta

Site selective C-H functionalization of Mitragyna alkaloids reveals a molecular switch for tuning opioid receptor signaling efficacy

帽柱木碱的位点选择性CH官能化揭示了一种调节阿片受体信号传导效力的分子开关

Bhowmik, Srijita; Galeta, Juraj; Havel, Václav; Nelson, Melissa; Faouzi, Abdelfattah; Bechand, Benjamin; Ansonoff, Mike; Fiala, Tomas; Hunkele, Amanda; Kruegel, Andrew C; Pintar, John E; Majumdar, Susruta; Javitch, Jonathan A; Sames, Dalibor

Correction to: Mu Opioids Induce Biased Signaling at the Full-Length Seven Transmembrane C-Terminal Splice Variants of the mu Opioid Receptor Gene, Oprm1

更正:μ阿片受体在μ阿片受体基因Oprm1的全长七次跨膜C端剪接变体处诱导偏向性信号传导

Narayan, Ankita; Hunkele, Amanda; Xu, Jin; Bassoni, Daniel L; Pasternak, Gavril W; Pan, Ying-Xian

Alternatively spliced mu opioid receptor C termini impact the diverse actions of morphine

μ阿片受体C端选择性剪接影响吗啡的多种作用

Xu, Jin; Lu, Zhigang; Narayan, Ankita; Le Rouzic, Valerie P; Xu, Mingming; Hunkele, Amanda; Brown, Taylor G; Hoefer, William F; Rossi, Grace C; Rice, Richard C; Martínez-Rivera, Arlene; Rajadhyaksha, Anjali M; Cartegni, Luca; Bassoni, Daniel L; Pasternak, Gavril W; Pan, Ying-Xian