High-throughput diversification of protein-ligand surfaces to discover chemical inducers of proximity
利用高通量方法对蛋白质-配体表面进行多样化修饰,以发现邻近效应的化学诱导剂。
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影响因子:
doi:10.1101/2024.09.30.615685
Shaum, James B; Muñoz I Ordoño, Miquel; Steen, Erica A; Wenge, Daniela V; Cheong, Hakyung; Hunkeler, Moritz; Bilotta, Eric M; Rutter, Zoe; Barta, Paige A; Thornhill, Abby M; Milosevich, Natalia; Hargis, Lauren M; Janowski, Jordan; Bishop, Timothy R; Carter, Trever R; da Camara, Bryce; Hinterndorfer, Matthias; Dada, Lucas; He, Wen-Ji; Offensperger, Fabian; Furihata, Hirotake; Schweber, Sydney R; Hatton, Charlie; Wen, Yanhe; Cravatt, Benjamin F; Engle, Keary M; Donovan, Katherine A; Melillo, Bruno; Kitamura, Seiya; Ciulli, Alessio; Armstrong, Scott A; Fischer, Eric S; Winter, Georg E; Erb, Michael A