日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

USP2 inhibition prevents infection with ACE2-dependent coronaviruses in vitro and is protective against SARS-CoV-2 in mice

USP2 抑制可在体外预防 ACE2 依赖性冠状病毒感染,并可在小鼠体内预防 SARS-CoV-2

Fabin Dang, Lei Bai, Jiazhen Dong, Xiaoping Hu, Jingchao Wang, Joao A Paulo, Yan Xiong, Xiaowei Liang, Yishuang Sun, Yuncai Chen, Ming Guo, Xin Wang, Zhixiang Huang, Hiroyuki Inuzuka, Li Chen, Chen Chu, Jianping Liu, Tao Zhang, Abdol-Hossein Rezaeian, Jing Liu, Husnu Ümit Kaniskan, Bo Zhong, Jinfang

De Novo Design of κ-Opioid Receptor Antagonists Using a Generative Deep-Learning Framework

利用生成式深度学习框架从头设计κ-阿片受体拮抗剂

Salas-Estrada, Leslie; Provasi, Davide; Qiu, Xing; Kaniskan, Husnu Ümit; Huang, Xi-Ping; DiBerto, Jeffrey F; Lamim Ribeiro, João Marcelo; Jin, Jian; Roth, Bryan L; Filizola, Marta

Targeted Degradation of PRC1 Components, BMI1 and RING1B, via a Novel Protein Complex Degrader Strategy

通过新型蛋白质复合物降解剂策略靶向降解 PRC1 成分 BMI1 和 RING1B

Kwang-Su Park, Lihuai Qin, Md Kabir, Kaixiu Luo, Brandon Dale, Yue Zhong, Arum Kim, Gang Greg Wang, Husnu Ümit Kaniskan, Jian Jin