日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Backbone Protecting Groups for Enhanced Peptide and Protein Synthesis

用于增强肽和蛋白质合成的骨架保护基团

Paravizzini, Samuel J; Haugaard-Kedström, Linda M; Hutton, Craig A; Karas, John A

Tetrahydropyranyl Backbone Protection for Enhanced Fmoc Solid-Phase Peptide Synthesis

四氢吡喃骨架保护增强Fmoc固相肽合成

Paravizzini, Samuel J; Hutton, Craig A; Karas, John A

A potent and selective reaction hijacking inhibitor of Plasmodium falciparum tyrosine tRNA synthetase exhibits single dose oral efficacy in vivo.

一种强效且选择性的恶性疟原虫酪氨酸 tRNA 合成酶反应劫持抑制剂在体内表现出单剂量口服疗效

Xie Stanley C, Tai Chia-Wei, Morton Craig J, Ma Liting, Huang Shih-Chung, Wittlin Sergio, Du Yawei, Hu Yongbo, Dogovski Con, Salimimarand Mina, Griffin Robert, England Dylan, de la Cruz Elisa, Deni Ioanna, Yeo Tomas, Burkhard Anna Y, Striepen Josefine, Schindler Kyra A, Crespo Benigno, Gamo Francisco J, Khandokar Yogesh, Hutton Craig A, Rabie Tayla, Birkholtz Lyn-Marié, Famodimu Mufuliat T, Delves Michael J, Bolsher Judith, Koolen Karin M J, van der Laak Rianne, Aguiar Anna C C, Pereira Dhelio B, Guido Rafael V C, Creek Darren J, Fidock David A, Dick Lawrence R, Brand Stephen L, Gould Alexandra E, Langston Steven, Griffin Michael D W, Tilley Leann

Site Specific Preparation of N-Glycosylated Peptides: Thioamide-Directed Activation of Aspartate

位点特异性制备N-糖基化肽:硫酰胺导向的天冬氨酸活化

Taresh, Ameer B; Hutton, Craig A

Effective Preparation of [(18)F]Flumazenil Using Copper-Mediated Late-Stage Radiofluorination of a Stannyl Precursor

利用铜介导的锡基前体后期放射性氟化反应高效制备[(18)F]氟马西尼

Haskali, Mohammad B; Roselt, Peter D; O'Brien, Terence J; Hutton, Craig A; Ali, Idrish; Vivash, Lucy; Jupp, Bianca

4-Nitrophenyl activated esters are superior synthons for indirect radiofluorination of biomolecules

4-硝基苯基活化酯是生物分子间接放射性氟化反应的优良合成子。

Haskali, Mohammad B; Farnsworth, Ashleigh L; Roselt, Peter D; Hutton, Craig A

Automated preparation of clinical grade [(68)Ga]Ga-DOTA-CP04, a cholecystokinin-2 receptor agonist, using iPHASE MultiSyn synthesis platform

利用iPHASE MultiSyn合成平台自动制备临床级胆囊收缩素-2受体激动剂[(68)Ga]Ga-DOTA-CP04

Haskali, Mohammad B; Roselt, Peter D; Binns, David; Hetsron, Amit; Poniger, Stan; Hutton, Craig A; Hicks, Rodney J

Hormetic potential of methylglyoxal, a side-product of glycolysis, in switching tumours from growth to death.

甲基乙二醛是糖酵解的副产物,它具有促进肿瘤从生长转变为死亡的激素效应

Nokin Marie-Julie, Durieux Florence, Bellier Justine, Peulen Olivier, Uchida Koji, Spiegel David A, Cochrane James R, Hutton Craig A, Castronovo Vincent, Bellahcène Akeila

Crystallization and preliminary X-ray diffraction analysis of diaminopimelate epimerase from Escherichia coli

大肠杆菌二氨基庚二酸差向异构酶的结晶和初步X射线衍射分析

Hor, Lilian; Dobson, Renwick C J; Dogovski, Con; Hutton, Craig A; Perugini, Matthew A

Expression, purification, crystallization and preliminary X-ray diffraction analysis of dihydrodipicolinate synthase from Bacillus anthracis in the presence of pyruvate

在丙酮酸存在下,炭疽芽孢杆菌二氢吡啶二羧酸合成酶的表达、纯化、结晶及初步X射线衍射分析

Voss, Jarrod E; Scally, Stephen W; Taylor, Nicole L; Dogovski, Con; Alderton, Malcolm R; Hutton, Craig A; Gerrard, Juliet A; Parker, Michael W; Dobson, Renwick C J; Perugini, Matthew A