Thiol-Reactive or Redox-Active: Revising a Repurposing Screen Led to a New Invalidation Pipeline and Identified a True Noncovalent Inhibitor Against Papain-like Protease from SARS-CoV-2.
硫醇反应性或氧化还原活性:修改重新定位筛选导致新的无效化流程,并鉴定出针对 SARS-CoV-2 木瓜蛋白酶样蛋白酶的真正非共价抑制剂
期刊:ACS Pharmacology and Translational Science
影响因子:3.7
doi:10.1021/acsptsci.4c00325
Kuzikov Maria, Morasso Stefano, Reinshagen Jeanette, Wolf Markus, Monaco Vittoria, Cozzolino Flora, GoliÄ Grdadolnik Simona, Å ket Primož, Plavec Janez, Iaconis Daniela, Summa Vincenzo, Corona Angela, Paulis Annalaura, Esposito Francesca, Tramontano Enzo, Monti Maria, Beccari Andrea R, Manelfi Candida, Windshügel Björn, Gribbon Philip, Storici Paola, Zaliani Andrea