日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Selective STING Activation in Intratumoral Myeloid Cells via CCR2-Directed Antibody-Drug Conjugate TAK-500

通过 CCR2 靶向抗体药物偶联物 TAK-500 选择性激活肿瘤内髓系细胞中的 STING

Vicky A Appleman ,Atsushi Matsuda ,Michelle L Ganno ,Dong Mei Zhang ,Emily Rosentrater ,Angel E Maldonado Lopez ,Angelo Porciuncula ,Tiquella Hatten ,Camilla L Christensen ,Samantha A Merrigan ,Hong Myung Lee ,Min Young Lee ,Charlotte I Wang ,Linlin Dong ,Jian Huang ,Natasha Iartchouk ,Jianing Wang ,He Xu ,Tomoki Yoneyama ,Konstantin I Piatkov ,Satyajeet Haridas ,Carole E Harbison ,Richard C Gregory ,Alexander Parent ,Neil Lineberry ,Chris Arendt ,Kurt A Schalper ,Adnan O Abu-Yousif

Genomic crosstalk between carbachol, a muscarinic receptor agonist, and the long-acting β(2)-adrenoceptor agonist, indacaterol, in human airway epithelial cells.

卡巴胆碱(一种毒蕈碱受体激动剂)与长效β2-肾上腺素受体激动剂茚达特罗在人类呼吸道上皮细胞中的基因组串扰

Jayasinghe Varuna, Joshi Radhika, Joshi Taruna, Paracha Tamkeen U, Kooi Cora, Mostafa Mahmoud M, Bauer Carla M T, Charlton Steven J, Iartchouk Oleg, Maillet Ashley, Morris Melody K, Ruda Vera M, Sandham David A, Wang Yanqun, Newton Robert, Giembycz Mark A

SHP2 blockade enhances anti-tumor immunity via tumor cell intrinsic and extrinsic mechanisms

SHP2阻断通过肿瘤细胞内在和外在机制增强抗肿瘤免疫力。

Ye Wang ,Morvarid Mohseni ,Angelo Grauel ,Javier Estrada Diez ,Wei Guan ,Simon Liang ,Jiyoung Elizabeth Choi ,Minying Pu ,Dongshu Chen ,Tyler Laszewski ,Stephanie Schwartz ,Jane Gu ,Leandra Mansur ,Tyler Burks ,Lauren Brodeur ,Roberto Velazquez ,Steve Kovats ,Bhavesh Pant ,Giri Buruzula ,Emily Deng ,Julie T Chen ,Farid Sari-Sarraf ,Christina Dornelas ,Malini Varadarajan ,Haiyan Yu ,Chen Liu ,Joanne Lim ,Huai-Xiang Hao ,Xiaomo Jiang ,Anthony Malamas ,Matthew J LaMarche ,Felipe Correa Geyer ,Margaret McLaughlin ,Carlotta Costa ,Joel Wagner ,David Ruddy ,Pushpa Jayaraman ,Nathaniel D Kirkpatrick ,Pu Zhang ,Oleg Iartchouk ,Kimberly Aardalen ,Viviana Cremasco ,Glenn Dranoff ,Jeffrey A Engelman ,Serena Silver ,Hongyun Wang ,William D Hastings # ,Silvia Goldoni #

TGFβ-blockade uncovers stromal plasticity in tumors by revealing the existence of a subset of interferon-licensed fibroblasts

TGFβ阻断揭示了肿瘤基质的可塑性,表现为存在一类经干扰素激活的成纤维细胞。

Angelo L Grauel ,Beverly Nguyen ,David Ruddy ,Tyler Laszewski ,Stephanie Schwartz ,Jonathan Chang ,Julie Chen ,Michelle Piquet ,Marc Pelletier ,Zheng Yan ,Nathaniel D Kirkpatrick ,Jincheng Wu ,Antoine deWeck ,Markus Riester ,Matt Hims ,Felipe Correa Geyer ,Joel Wagner ,Kenzie MacIsaac ,James Deeds ,Rohan Diwanji ,Pushpa Jayaraman ,Yenyen Yu ,Quincey Simmons ,Shaobu Weng ,Alina Raza ,Brian Minie ,Mirek Dostalek ,Pavitra Chikkegowda ,Vera Ruda ,Oleg Iartchouk ,Naiyan Chen ,Raphael Thierry ,Joseph Zhou ,Iulian Pruteanu-Malinici ,Claire Fabre ,Jeffrey A Engelman ,Glenn Dranoff ,Viviana Cremasco

Target (MexB)- and Efflux-Based Mechanisms Decreasing the Effectiveness of the Efflux Pump Inhibitor D13-9001 in Pseudomonas aeruginosa PAO1: Uncovering a New Role for MexMN-OprM in Efflux of β-Lactams and a Novel Regulatory Circuit (MmnRS) Controlling MexMN Expression

靶向(MexB)和外排机制降低铜绿假单胞菌PAO1中外排泵抑制剂D13-9001的有效性:揭示MexMN-OprM在β-内酰胺类抗生素外排中的新作用以及控制MexMN表达的新型调控回路(MmnRS)

Ranjitkar, Srijan; Jones, Adriana K; Mostafavi, Mina; Zwirko, Zachary; Iartchouk, Oleg; Barnes, S Whitney; Walker, John R; Willis, Thomas W; Lee, Patrick S; Dean, Charles R

Short-term Low-Dose mTORC1 Inhibition in Aged Rats Counter-Regulates Age-Related Gene Changes and Blocks Age-Related Kidney Pathology

短期低剂量抑制老年大鼠的 mTORC1 可反调节与年龄相关的基因变化并阻止与年龄相关的肾脏病理

Tea Shavlakadze, Jiang Zhu, Sharon Wang, Weihua Zhou, Bret Morin, Marc A Egerman, Lin Fan, Yanqun Wang, Oleg Iartchouk, Angelika Meyer, Reginald A Valdez, Joan B Mannick, Lloyd B Klickstein, David J Glass

Genetic Determinants of Drug Resistance in Mycobacterium tuberculosis and Their Diagnostic Value

结核分枝杆菌耐药性的遗传决定因素及其诊断价值

Farhat, Maha R; Sultana, Razvan; Iartchouk, Oleg; Bozeman, Sam; Galagan, James; Sisk, Peter; Stolte, Christian; Nebenzahl-Guimaraes, Hanna; Jacobson, Karen; Sloutsky, Alexander; Kaur, Devinder; Posey, James; Kreiswirth, Barry N; Kurepina, Natalia; Rigouts, Leen; Streicher, Elizabeth M; Victor, Tommie C; Warren, Robin M; van Soolingen, Dick; Murray, Megan

Highly multiplexed molecular inversion probe genotyping: over 10,000 targeted SNPs genotyped in a single tube assay

高通量分子反转探针基因分型:单管检测即可完成超过10,000个靶向SNP的基因分型

Hardenbol, Paul; Yu, Fuli; Belmont, John; Mackenzie, Jennifer; Bruckner, Carsten; Brundage, Tiffany; Boudreau, Andrew; Chow, Steve; Eberle, Jim; Erbilgin, Ayca; Falkowski, Mat; Fitzgerald, Ron; Ghose, Sy; Iartchouk, Oleg; Jain, Maneesh; Karlin-Neumann, George; Lu, Xiuhua; Miao, Xin; Moore, Bridget; Moorhead, Martin; Namsaraev, Eugeni; Pasternak, Shiran; Prakash, Eunice; Tran, Karen; Wang, Zhiyong; Jones, Hywel B; Davis, Ronald W; Willis, Thomas D; Gibbs, Richard A