日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of AZD4144, a Selective and Potent NLRP3 Inhibitor for the Treatment of Inflammatory Diseases.

发现 AZD4144,一种选择性强效的 NLRP3 抑制剂,可用于治疗炎症性疾病

Johansson Anders, Sugama Hiroshi, Larsson Niklas, Winiwarter Susanne, Yoshida Kosuke, Gradén Henrik, Bergonzini Giulia, Matsumura Takehiko, Miyazaki Shiki, Fuchigami Ryuichi, Eda Masahiro, Takamatsu Hisayuki, Iguchi Kaori, Hongu Mitsuya, Matsudaira Tetsuji, Hovdal Daniel, Fredenwall Marlene, Fahlander Ulf, Luchniak Anna, Brengdahl Johan, Jung Bomi, Rhedin Magdalena, Sardana Juhi, Idei Akiko, Kato Yosuke, Kimura Junpei, Viklund Jenny, Brandt Peter, Sjögren Anna-Karin, Hibino Yui, Woollard Kevin, Yoneda Hikaru

Discovery of a novel class NSD2 inhibitor for multiple myeloma with t(4;14)().

发现一种新型 NSD2 抑制剂,用于治疗伴有 t(4;14) 的多发性骨髓瘤。

Matsuoka Sae, Osada Naoki, Kubota Hirokazu, Kikuzato Ko, Koyama Hiroo, Sonoda Takeshi, Idei Akiko, Yoshida Minoru, Kikuchi Masaki, Umehara Takashi, Watanabe Chiduru, Honma Teruki, Yasui Hiroshi, Ikeda Sho, Takahashi Naoto, Nakasone Hideki, Kikuchi Jiro, Furukawa Yusuke

Synergistic involvement of the NZF domains of the LUBAC accessory subunits HOIL-1L and SHARPIN in the regulation of LUBAC function

LUBAC辅助亚基HOIL-1L和SHARPIN的NZF结构域协同参与LUBAC功能的调控

Toda, Yusuke; Fujita, Hiroaki; Mino, Koshiki; Koyama, Takuto; Matsuoka, Seiji; Kaizuka, Toshie; Agawa, Mari; Matsumoto, Shigeyuki; Idei, Akiko; Nishikori, Momoko; Okuno, Yasushi; Osada, Hiroyuki; Yoshida, Minoru; Takaori-Kondo, Akifumi; Iwai, Kazuhiro