Rational Design of Dual-Domain Binding Inhibitors for N-Acetylgalactosamine Transferase 2 with Improved Selectivity over the T1 and T3 Isoforms
合理设计对N-乙酰半乳糖胺转移酶2具有更高选择性的双结构域结合抑制剂(针对T1和T3亚型)
期刊:JACS Au
影响因子:8.7
doi:10.1021/jacsau.4c00633
Compañón, Ismael; Ballard, Collin J; Lira-Navarrete, Erandi; Santos, Tanausú; Monaco, Serena; Muñoz-García, Juan C; Delso, Ignacio; Angulo, Jesus; Gerken, Thomas A; Schjoldager, Katrine T; Clausen, Henrik; Tejero, Tomás; Merino, Pedro; Corzana, Francisco; Hurtado-Guerrero, Ramon; Ghirardello, Mattia