日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of Hantzsch Adducts as Cholinesterases and Calcium Flux inhibitors, Antioxidants and Neuroprotectives

Hantzsch 加合物作为胆碱酯酶和钙通量抑制剂、抗氧化剂和神经保护剂的合成

Irene Pachón Angona, Helene Martin, Solene Daniel, Ignacio Moraleda, Alexandre Bonet, Artur Wnorowski, Maciej Maj, Krzysztof Jozwiak, Isabel Iriepa, Bernard Refouvelet, José Marco-Contelles, Lhassane Ismaili

Imidazopyranotacrines as Non-Hepatotoxic, Selective Acetylcholinesterase Inhibitors, and Antioxidant Agents for Alzheimer's Disease Therapy

咪唑并吡喃他克林作为无肝毒性、选择性乙酰胆碱酯酶抑制剂和抗氧化剂用于治疗阿尔茨海默病

Houssem Boulebd, Lhassane Ismaili, Manuela Bartolini, Abdelmalek Bouraiou, Vincenza Andrisano, Helene Martin, Alexandre Bonet, Ignacio Moraleda, Isabel Iriepa, Mourad Chioua, Ali Belfaitah, José Marco-Contelles2

Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer's disease: design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybrids

用于治疗阿尔茨海默病的多效胆碱酯酶/单胺氧化酶抑制剂:新型多奈哌齐-吡啶杂化物的设计、合成、生化评价、ADMET、分子建模和 QSAR 分析

Oscar M Bautista-Aguilera, Gerard Esteban, Mourad Chioua, Katarina Nikolic, Danica Agbaba, Ignacio Moraleda, Isabel Iriepa, Elena Soriano, Abdelouahid Samadi, Mercedes Unzeta, José Marco-Contelles

Synthesis, pharmacological assessment, and molecular modeling of acetylcholinesterase/butyrylcholinesterase inhibitors: effect against amyloid-β-induced neurotoxicity

乙酰胆碱酯酶/丁酰胆碱酯酶抑制剂的合成、药理学评估和分子建模:对抗淀粉样蛋白-β诱导的神经毒性的作用

Daniel Silva, Mourad Chioua, Abdelouahid Samadi, Paula Agostinho, Pedro Garção, Rocío Lajarín-Cuesta, Cristobal de Los Ríos, Isabel Iriepa, Ignacio Moraleda, Laura Gonzalez-Lafuente, Eduarda Mendes, Concepción Pérez, María Isabel Rodríguez-Franco, José Marco-Contelles, M Carmo Carreiras