日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Comparative Study of Allosteric GPCR Binding Sites and Their Ligandability Potential

变构GPCR结合位点及其配体结合潜能的比较研究

Peter, Sonja; Siragusa, Lydia; Thomas, Morgan; Palomba, Tommaso; Cross, Simon; O'Boyle, Noel M; Bajusz, Dávid; Ferenczy, György G; Keserű, György M; Bottegoni, Giovanni; Bender, Brian; Chen, Ijen; De Graaf, Chris

Exploring IDP-Ligand Interactions: tau K18 as A Test Case

探索 IDP-配体相互作用:以 tau K18 为例

Darius Vagrys, James Davidson, Ijen Chen, Roderick E Hubbard, Ben Davis

Establishing Drug Discovery and Identification of Hit Series for the Anti-apoptotic Proteins, Bcl-2 and Mcl-1

建立抗凋亡蛋白 Bcl-2 和 Mcl-1 的药物发现和热门系列鉴定

James B Murray, James Davidson, Ijen Chen, Ben Davis, Pawel Dokurno, Christopher J Graham, Richard Harris, Allan Jordan, Natalia Matassova, Christopher Pedder, Stuart Ray, Stephen D Roughley, Julia Smith, Claire Walmsley, Yikang Wang, Neil Whitehead, Douglas S Williamson, Patrick Casara, Thierry Le

S55746 is a novel orally active BCL-2 selective and potent inhibitor that impairs hematological tumor growth

S55746 是一种新型口服 BCL-2 选择性强效抑制剂,可抑制血液肿瘤生长

Patrick Casara #, James Davidson #, Audrey Claperon #, Gaëtane Le Toumelin-Braizat, Meike Vogler, Alain Bruno, Maïa Chanrion, Gaëlle Lysiak-Auvity, Thierry Le Diguarher, Jérôme-Benoît Starck, Ijen Chen, Neil Whitehead, Christopher Graham, Natalia Matassova, Pawel Dokurno, Christopher Pedder, Youzhen