日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis of a Cannabidiol Precursor: Experimental Challenges and DFT Insights into β‑Elimination Barriers

大麻二酚前体的合成:实验挑战和DFT对β-消除能垒的见解

Bergami, Michael; Trapella, Claudio; Compagnin, Greta; Felletti, Simona; Catani, Martina; Pezzola, Silvia; Sabuzi, Federica; Galloni, Pierluca; Marchetti, Paolo; Cristofori, Virginia; Fantinati, Anna; Illuminati, Davide

Synthesis and Pharmacological Characterization of Nociceptin/Orphanin FQ Dimeric Ligands

伤害感受素/孤啡肽FQ二聚体配体的合成及药理学表征

Albanese, Valentina; Pola, Pietro; Argentieri, Michela; De Ventura, Tiziano; Frezza, Alessia; Illuminati, Davide; Malfacini, Davide; Marzola, Erika; Meneguzzo, Giulio; Morrone, Erika; Preti, Delia; Rizzo, Alessandra; Sturaro, Chiara; Calò, Girolamo; Guerrini, Remo; Pacifico, Salvatore; Ruzza, Chiara

Multi-Step Synthesis of Chimeric Nutlin-DCA Compounds Targeting Dual Pathways for Treatment of Cancer

利用多步合成法合成靶向双重通路的嵌合型Nutlin-DCA化合物用于癌症治疗

Illuminati, Davide; Foschi, Rebecca; Marchetti, Paolo; Zanirato, Vinicio; Fantinati, Anna; Trapella, Claudio; Voltan, Rebecca; Cristofori, Virginia

Spiropiperidine-Based Oligomycin-Analog Ligands To Counteract the Ischemia-Reperfusion Injury in a Renal Cell Model

基于螺哌啶的寡霉素类似物配体在肾细胞模型中对抗缺血再灌注损伤

Turrin, Giulia; Lo Cascio, Ettore; Giacon, Noah; Fantinati, Anna; Cristofori, Virginia; Illuminati, Davide; Preti, Delia; Morciano, Giampaolo; Pinton, Paolo; Agyapong, Esther Densu; Trapella, Claudio; Arcovito, Alessandro

Methyl-Containing Pharmaceuticals

含甲基药物

Illuminati, Davide; Fantinati, Anna

Enhanced anticancer effect of thymidylate synthase dimer disrupters by promoting intracellular accumulation.

胸苷酸合成酶二聚体破坏剂通过促进细胞内积累增强抗癌作用

Marverti Gaetano, Moschella Maria Gaetana, Belardo Alice, Lamesta Michele, Mercanile Giada, Tagliazucchi Lorenzo, Aiello Daniele, Venturelli Alberto, Illuminati Davide, Guerrini Remo, Losi Lorena, Ponterini Glauco, Costi Maria Paola, D'Arca Domenico

Enzymatic Desymmetrisation of Prochiral meso-1,2-Disubstituted-1,2-Diaminoethane for the Synthesis of Key Enantioenriched (-)-Nutlin-3 Precursor

利用酶促去对称化反应合成关键的对映体富集的(-)-Nutlin-3前体,以合成前手性内消旋-1,2-二取代-1,2-二氨基乙烷。

Cristofori, Virginia; Illuminati, Davide; Bisquoli, Chiara; Catani, Martina; Compagnin, Greta; Turrin, Giulia; Trapella, Claudio; Fantinati, Anna

(L)-Monomethyl Tyrosine (Mmt): New Synthetic Strategy via Bulky 'Forced-Traceless' Regioselective Pd-Catalyzed C(sp(2))-H Activation

(L)-单甲基酪氨酸 (Mmt):通过大位阻“强制无痕”区域选择性钯催化C(sp(2))-H活化实现的新合成策略

Illuminati, Davide; Trapella, Claudio; Zanirato, Vinicio; Guerrini, Remo; Albanese, Valentina; Sturaro, Chiara; Stragapede, Simona; Malfacini, Davide; Compagnin, Greta; Catani, Martina; Fantinati, Anna

Novel Mixed NOP/Opioid Receptor Peptide Agonists

新型混合型NOP/阿片受体肽激动剂

Pacifico, Salvatore; Albanese, Valentina; Illuminati, Davide; Marzola, Erika; Fabbri, Martina; Ferrari, Federica; Holanda, Victor A D; Sturaro, Chiara; Malfacini, Davide; Ruzza, Chiara; Trapella, Claudio; Preti, Delia; Lo Cascio, Ettore; Arcovito, Alessandro; Della Longa, Stefano; Marangoni, Martina; Fattori, Davide; Nassini, Romina; Calò, Girolamo; Guerrini, Remo