日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Phosphoinositide-dependent kinase 1 (PDK1) in cancer: molecular insights and therapeutic strategies

癌症中的磷脂酰肌醇依赖性激酶1 (PDK1):分子机制及治疗策略

Algheribe, Shatha; Zagzoog, Ayat; Boudjelal, Mohamed; Islam, Imadul

Novel benzimidazole-1, 3, 4-thiadiazole derivatives as casein kinase-2 inhibitors: synthesis, in vitro and in silico investigations

新型苯并咪唑-1,3,4-噻二唑衍生物作为酪蛋白激酶-2抑制剂:合成、体外和计算机模拟研究

Senthilkumar, N; Sarveswari, S; Choudhari, Prafulla; Chaudhari, Somdatta; Islam, Imadul; Tamboli, Yasinalli; Vijayakumar, V

First-in-class inhibitors of Nsp15 endoribonuclease of SARS-CoV-2: Modeling, synthesis, and enzymatic assay of thiazolidinedione and rhodanine analogs

SARS-CoV-2 Nsp15 核糖核酸内切酶的首创抑制剂:噻唑烷二酮和罗丹宁类似物的建模、合成和酶活性测定

Mehyar, Nimer; Samman, Nosaibah; Al Gheribi, Shatha; Mashhour, Abdullah; Chan, Pearl; Al-Kaysi, Rabih O; Perlman, Stanley; Boudjelal, Mohamed; Islam, Imadul

Genomics-driven drug repurposing and novel targets identification for sickle cell disease in Saudi patients

基因组学驱动的药物再利用和新靶点识别在沙特阿拉伯镰状细胞病患者中的应用

Alghubayshi, Ali; Alshabeeb, Mohammad A; Wijesinghe, Dayanjan; AlAwadh, Mohammed; Alshammari, Suad; Alrajeh, Khalifa; Alkhairi, Mona A; Islam, Imadul; Alaskar, Ahmed

Therapeutic drug monitoring of busulfan in pediatric patients: a 5-year observational study

儿童患者使用白消安进行治疗药物监测:一项为期5年的观察性研究

Alomari, Nedaa; Kurdi, Amani; Alghamdi, Meshari; Alhussaini, Waleed; Ezzeldeen, Ghanem; Alharbi, Eman; Aldahri, Alaa; Islam, Imadul; Essa, Mohammed

Novel 2,4-Dichloro-5-sulfamoylbenzoic Acid Oxime Esters: First Studies as Potential Human Carbonic Anhydrase Inhibitors

新型2,4-二氯-5-氨磺酰基苯甲酸肟酯:作为潜在的人类碳酸酐酶抑制剂的初步研究

Kilbile, Jaydeo T; Sapkal, Suryakant B; Renzi, Gioele; D'Agostino, Ilaria; Cutarella, Luigi; Mori, Mattia; De Filippis, Barbara; Islam, Imadul; Massardi, Maria Luisa; Somenza, Elena; Ronca, Roberto; Tamboli, Yasinalli; Carta, Fabrizio; Supuran, Claudiu T

Comparative performance of liquid chromatography and spectrophotometry in determining metformin hydrochloride within pharmaceutical formulations

液相色谱法和分光光度法测定药物制剂中的盐酸二甲双胍的比较性能

Amani Kurdi, Waleed Alhussaini, Abdulrahman Alawaji, Abdullah Alhudathi, Rakan Alharbi, Faisal Binsaleh, Yazeed Alghamidi, Abdulkareem Al Bekairy, Abdulmalik Alkatheri, Imadul Islam, Ibrahim Farh, Ezzeldeen Ghanem, Mahmoud Mansour

First Report from Saudi Arabia of Trimethylaminuria Caused by a Premature Stop Codon Mutation in the FMO3 Gene

沙特阿拉伯首次报道由FMO3基因提前终止密码子突变引起的三甲胺尿症

Alghanem, Bandar; Alamri, Hassan S; Barhoumi, Tlili; Ali Khan, Imran; Almuhalhil, Khawlah; Aloyouni, Essra; Shaibah, Hayat; Mashhour, Abdullah; Algheribe, Shatha; Islam, Imadul; Boudjelal, Mohamed; Alfadhel, Majid

Distinct Mechanisms of Cytotoxicity in Novel Nitrogenous Heterocycles: Future Directions for a New Anti-Cancer Agent

新型含氮杂环化合物独特的细胞毒性机制:新型抗癌药物的未来发展方向

Suliman, Rasha Saad; Alghamdi, Sahar Saleh; Ali, Rizwan; Rahman, Ishrat; Alqahtani, Tariq; Frah, Ibrahim K; Aljatli, Dimah A; Huwaizi, Sarah; Algheribe, Shatha; Alehaideb, Zeyad; Islam, Imadul

Therapeutics discovery: From bench to first in-human trials

治疗药物发现:从实验室到首次人体试验

Al-Hujaily, Ensaf M; Khatlani, Tanvir; Alehaideb, Zeyad; Ali, Rizwan; Almuzaini, Bader; Alrfaei, Bahauddeen M; Iqbal, Jahangir; Islam, Imadul; Malik, Shuja; Marwani, Bader A; Massadeh, Salam; Nehdi, Atef; Alsomaie, Barrak; Debasi, Bader; Bushnak, Ibraheem; Noibi, Saeed; Hussain, Syed; Wajid, Wahid Abdul; Armand, Jean-Pierre; Gul, Sheraz; Oyarzabal, Julen; Rais, Rana; Bountra, Chas; Alaskar, Ahmed; Knawy, Bander Al; Boudjelal, Mohamed