Trivalent PROTACs enhance protein degradation via combined avidity and cooperativity
三价 PROTAC 通过结合亲和力和协同作用增强蛋白质降解
期刊:Nature Chemical Biology
影响因子:12.9
doi:10.1038/s41589-021-00878-4
Satomi Imaide #, Kristin M Riching #, Nikolai Makukhin #, Vesna Vetma, Claire Whitworth, Scott J Hughes, Nicole Trainor, Sarah D Mahan, Nancy Murphy, Angus D Cowan, Kwok-Ho Chan, Conner Craigon, Andrea Testa, Chiara Maniaci, Marjeta Urh, Danette L Daniels, Alessio Ciulli