日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Rogocekib (CTX-712): A Potent and Selective CLK Inhibitor for Cancer Treatment

罗戈西克布(CTX-712)的发现:一种强效且选择性的CLK抑制剂,可用于癌症治疗

Kawakita, Youichi; Kojima, Takuto; Nii, Noriyuki; Ito, Yoshiteru; Sakauchi, Nobuki; Banno, Hiroshi; Liu, Xin; Ono, Koji; Imamura, Keisuke; Imamura, Shinichi; Iwai, Kenichi; Yamamoto, Yukiko; Iwatani, Misa; Uchiyama, Noriko; Sugiyama, Midori; Mizutani, Akio; Satoh, Yoshihiko; Arikawa, Yasuyoshi; Morishita, Daisuke; Shimokawa, Kenichiro

Evaluation of specific binding of [(11)C]TZ7774 to the receptor-interacting protein kinase 1 (RIPK1) in the brain

评估[(11)C]TZ7774与脑内受体相互作用蛋白激酶1 (RIPK1)的特异性结合

Sakai, Takayuki; Yamada, Takashi; Ikenuma, Hiroshi; Ogata, Aya; Ichise, Masanori; Hattori, Saori; Abe, Junichiro; Tada, Mari; Kakita, Akiyoshi; Suzuki, Masaaki; Ito, Kengo; Kato, Takashi; Imamura, Shinichi; Kimura, Yasuyuki

Anti-angiogenic and anti-tumor effects of TAK-593, a potent and selective inhibitor of vascular endothelial growth factor and platelet-derived growth factor receptor tyrosine kinase.

TAK-593 是一种强效且选择性的血管内皮生长因子和血小板衍生生长因子受体酪氨酸激酶抑制剂,具有抗血管生成和抗肿瘤作用

Awazu Yoshiko, Mizutani Akio, Nagase Yoshinori, Tsuchiya Shuntarou, Nakamura Kazuhide, Kakoi Yuichi, Kitahara Osamu, Takeuchi Toshiyuki, Yamasaki Seiji, Miyamoto Naoki, Iwata Hidehisa, Miki Hiroshi, Imamura Shinichi, Hori Akira

A novel pyrrolo[3, 2-d]pyrimidine derivative, as a vascular endothelial growth factor receptor and platelet-derived growth factor receptor tyrosine kinase inhibitor, shows potent antitumor activity by suppression of tumor angiogenesis.

一种新型吡咯并[3, 2-d]嘧啶衍生物,作为血管内皮生长因子受体和血小板衍生生长因子受体酪氨酸激酶抑制剂,通过抑制肿瘤血管生成显示出强大的抗肿瘤活性

Awazu Yoshiko, Mizutani Akio, Nagase Yoshinori, Iwata Hidehisa, Oguro Yuya, Miki Hiroshi, Imamura Shinichi, Hori Akira

FOXA1 promotes tumor progression in prostate cancer via the insulin-like growth factor binding protein 3 pathway

FOXA1 通过胰岛素样生长因子结合蛋白 3 通路促进前列腺癌肿瘤进展

Yusuke Imamura, Shinichi Sakamoto, Takumi Endo, Takanobu Utsumi, Miki Fuse, Takahito Suyama, Koji Kawamura, Takashi Imamoto, Kojiro Yano, Katsuhiro Uzawa, Naoki Nihei, Hiroyoshi Suzuki, Atsushi Mizokami, Takeshi Ueda, Naohiko Seki, Hideki Tanzawa, Tomohiko Ichikawa

Chemotherapeutic evaluation of a synthetic tubulysin analogue-dendrimer conjugate in c26 tumor bearing mice

在荷瘤小鼠中对合成的微管溶素类似物-树状聚合物缀合物进行化疗评价

Floyd, William C 3rd; Datta, Gopal K; Imamura, Shinichi; Kieler-Ferguson, Heidi M; Jerger, Katherine; Patterson, Andrew W; Fox, Megan E; Szoka, Francis C; Fréchet, Jean M J; Ellman, Jonathan A

Fragment-based discovery of selective inhibitors of the Mycobacterium tuberculosis protein tyrosine phosphatase PtpA

基于片段的结核分枝杆菌蛋白酪氨酸磷酸酶 PtpA 选择性抑制剂的发现

Rawls, Katherine A; Lang, P Therese; Takeuchi, Jun; Imamura, Shinichi; Baguley, Tyler D; Grundner, Christoph; Alber, Tom; Ellman, Jonathan A