日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Based Design of New Series of Sulfonates with Potent and Specific BChE Inhibition and Anti-Inflammatory Effects

基于结构的新型磺酸盐系列设计及其强效和特异性的丁酰胆碱酯酶抑制和抗炎作用

Kurma, Siva Hariprasad; Adarvez-Feresin, Camila; Parravicini, Oscar; Garro, Adriana; Stepankova, Sarka; Hosek, Jan; Pauk, Karel; Lisicic, Jovana; Jampilek, Josef; Enriz, Ricardo Daniel; Imramovsky, Ales

Study of Biological Activities and ADMET-Related Properties of Salicylanilide-Based Peptidomimetics

水杨酰苯胺类肽模拟物的生物活性及ADMET相关特性研究

Dominika Pindjakova, Eliska Pilarova, Karel Pauk, Hana Michnova, Jan Hosek, Pratibha Magar, Alois Cizek, Ales Imramovsky, Josef Jampilek

SAR-mediated Similarity Assessment of the Property Profile for New, Silicon-Based AChE/BChE Inhibitors

SAR 介导的新型硅基 AChE/BChE 抑制剂特性相似性评估

Andrzej Bak, Hana Pizova, Violetta Kozik, Katarina Vorcakova, Jiri Kos, Jakub Treml, Klara Odehnalova, Michal Oravec, Ales Imramovsky, Pavel Bobal, Adam Smolinski, Zdeněk Trávníček, Josef Jampilek3

Novel Benzene-Based Carbamates for AChE/BChE Inhibition: Synthesis and Ligand/Structure-Oriented SAR Study

用于 AChE/BChE 抑制的新型苯基氨基甲酸酯:合成和配体/结构导向的 SAR 研究

Andrzej Bak, Violetta Kozik, Dariusz Kozakiewicz, Kamila Gajcy, Daniel Jan Strub, Aleksandra Swietlicka, Sarka Stepankova, Ales Imramovsky, Jaroslaw Polanski, Adam Smolinski, Josef Jampilek

Proline-Based Carbamates as Cholinesterase Inhibitors

脯氨酸基氨基甲酸酯作为胆碱酯酶抑制剂

Hana Pizova, Marketa Havelkova, Sarka Stepankova, Andrzej Bak, Tereza Kauerova, Violetta Kozik, Michal Oravec, Ales Imramovsky, Peter Kollar, Pavel Bobal, Josef Jampilek1

In vitro bactericidal activity of 4- and 5-chloro-2-hydroxy-N-[1-oxo-1-(phenylamino)alkan-2-yl]benzamides against MRSA

4-和5-氯-2-羟基-N-[1-氧代-1-(苯氨基)烷-2-基]苯甲酰胺对MRSA的体外杀菌活性

Iveta Zadrazilova, Sarka Pospisilova, Karel Pauk, Ales Imramovsky, Jarmila Vinsova, Alois Cizek, Josef Jampilek

Synthesis and antimycobacterial and photosynthesis-inhibiting evaluation of 2-[(E)-2-substituted-ethenyl]-1,3-benzoxazoles

2-[(E)-2-取代乙烯基]-1,3-苯并恶唑的合成及其抗分枝杆菌和光合作用抑制活性评价

Imramovsky, Ales; Kozic, Jan; Pesko, Matus; Stolarikova, Jirina; Vinsova, Jarmila; Kralova, Katarina; Jampilek, Josef

Antimycobacterial and photosynthetic electron transport inhibiting activity of ring-substituted 4-arylamino-7-chloroquinolinium chlorides

环取代的4-芳氨基-7-氯喹啉氯化物的抗分枝杆菌和光合电子传递抑制活性

Jan Otevrel, Pavel Bobal, Iveta Zadrazilova, Rodney Govender, Matus Pesko, Stanislava Keltosova, Petra Koleckarova, Petr Marsalek, Ales Imramovsky, Aidan Coffey, Jim O'Mahony, Peter Kollar, Alois Cizek, Katarina Kralova, Josef Jampilek

Antibacterial and herbicidal activity of ring-substituted 2-hydroxynaphthalene-1-carboxanilides

环取代2-羟基萘-1-甲酰苯胺的抗菌和除草活性

Tomas Gonec, Jiri Kos, Iveta Zadrazilova, Matus Pesko, Rodney Govender, Stanislava Keltosova, Barbara Chambel, Diogo Pereira, Peter Kollar, Ales Imramovsky, Jim O'Mahony, Aidan Coffey, Alois Cizek, Katarina Kralova, Josef Jampilek

Investigating the spectrum of biological activity of substituted quinoline-2-carboxamides and their isosteres

研究取代的喹啉-2-甲酰胺及其电子等排体的生物活性谱

Tomas Gonec, Pavel Bobal, Josef Sujan, Matus Pesko, Jiahui Guo, Katarina Kralova, Lenka Pavlacka, Libor Vesely, Eva Kreckova, Jiri Kos, Aidan Coffey, Peter Kollar, Ales Imramovsky, Lukas Placek, Josef Jampilek