日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An overview of drug-induced sodium channel blockade and changes in cardiac conduction: Implications for drug safety

药物诱导的钠通道阻滞及心脏传导改变概述:对药物安全性的影响

Chaudhary, Khuram W; Clancy, Colleen E; Yang, Pei-Chi; Pierson, Jennifer B; Goldin, Alan L; Koerner, John E; Wisialowski, Todd A; Valentin, Jean-Pierre; Imredy, John P; Lagrutta, Armando; Authier, Simon; Kleiman, Robert; Sager, Philip T; Hoffmann, Peter; Pugsley, Michael K

Cross-site and cross-platform variability of automated patch clamp assessments of drug effects on human cardiac currents in recombinant cells.

药物对重组细胞中人类心脏电流影响的自动膜片钳评估的跨站点和跨平台变异性

Kramer James, Himmel Herbert M, Lindqvist Anders, Stoelzle-Feix Sonja, Chaudhary Khuram W, Li Dingzhou, Bohme Georg Andrees, Bridgland-Taylor Matthew, Hebeisen Simon, Fan Jingsong, Renganathan Muthukrishnan, Imredy John, Humphries Edward S A, Brinkwirth Nina, Strassmaier Tim, Ohtsuki Atsushi, Danker Timm, Vanoye Carlos, Polonchuk Liudmila, Fermini Bernard, Pierson Jennifer Beck, Gintant Gary

Corrigendum to "A systematic strategy for estimating hERG block potency and its implications in a new cardiac safety paradigm" [Toxicology and Applied Pharmacology volume 394C (2020) 114961]

对“评估 hERG 阻滞效力的系统策略及其在新的心脏安全范式中的意义”的更正[毒理学和应用药理学卷 394C (2020) 114961]

Ridder, Bradley J; Leishman, Derek J; Bridgland-Taylor, Matthew; Samieegohar, Mohammadreza; Han, Xiaomei; Wu, Wendy W; Randolph, Aaron; Tran, Phu; Sheng, Jiansong; Danker, Timm; Lindqvist, Anders; Konrad, Daniel; Hebeisen, Simon; Polonchuk, Liudmila; Gissinger, Evgenia; Renganathan, Muthukrishnan; Koci, Bryan; Wei, Haiyang; Fan, Jingsong; Levesque, Paul; Kwagh, Jae; Imredy, John; Zhai, Jin; Rogers, Marc; Humphries, Edward; Kirby, Robert; Stoelzle-Feix, Sonja; Brinkwirth, Nina; Rotordam, Maria Giustina; Becker, Nadine; Friis, Søren; Rapedius, Markus; Goetze, Tom A; Strassmaier, Tim; Okeyo, George; Kramer, James; Kuryshev, Yuri; Wu, Caiyun; Himmel, Herbert; Mirams, Gary R; Strauss, David G; Bardenet, Remi; Li, Zhihua

A systematic strategy for estimating hERG block potency and its implications in a new cardiac safety paradigm.

评估 hERG 阻滞效力的系统策略及其在新心脏安全范式中的意义

Ridder Bradley J, Leishman Derek J, Bridgland-Taylor Matthew, Samieegohar Mohammadreza, Han Xiaomei, Wu Wendy W, Randolph Aaron, Tran Phu, Sheng Jiansong, Danker Timm, Lindqvist Anders, Konrad Daniel, Hebeisen Simon, Polonchuk Liudmila, Gissinger Evgenia, Renganathan Muthukrishnan, Koci Bryan, Wei Haiyang, Fan Jingsong, Levesque Paul, Kwagh Jae, Imredy John, Zhai Jin, Rogers Marc, Humphries Edward, Kirby Robert, Stoelzle-Feix Sonja, Brinkwirth Nina, Rotordam Maria Giustina, Becker Nadine, Friis Søren, Rapedius Markus, Goetze Tom A, Strassmaier Tim, Okeyo George, Kramer James, Kuryshev Yuri, Wu Caiyun, Himmel Herbert, Mirams Gary R, Strauss David G, Bardenet Rémi, Li Zhihua