日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A fission yeast-based platform for nematode PDE inhibitor discovery

基于裂殖酵母的线虫PDE抑制剂发现平台

Bibeau, Sarah; Chen, Natalie; Sutoris, Hannah; Ly, Judy; Eberhard, Jeremy; Hubbell, Sara M; Banda, Eric; Povh, Esther; Anindya, Clianta S; Berwanger, Michael R; Sinise, Sarah E; Zhang, Xieyang; Morken, James P; Galande, Kranti K; Cote, Rick H; Dranchak, Patricia K; Inglese, James; Hoffman, Charles S

A general assay platform to study protein pharmacology using ligand-dependent structural dynamics.

利用配体依赖性结构动力学研究蛋白质药理学的通用检测平台

Ciulla Daniel A, Dranchak Patricia K, Aitha Mahesh, van Neer Renier H P, Shah Divia, Tharakan Ravi, Wilson Kelli M, Wang Yuhong, Braisted John C, Inglese James

Metabolic engineering and late-stage functionalization expand the chemical space of the antimalarial premarineosin A

代谢工程和后期功能化扩展了抗疟药普瑞马利尼奥辛A的化学空间。

McBride, Christina M; McCauley, Morgan; Harris, Natalia R; Amin, Sahar; Curtis, Brian J; Verhey-Henke, Linnea; Teklemichael, Awet A; Oliphant, Erin N; Dranchak, Patricia; Lev, Katherine L; Qu, Fengrui; Snodgrass, Harrison M; Lewis, Jared C; Inglese, James; Su, Xin-Zhuan; Pereira, Filipa; Sherman, David H

A Quantitative High-Throughput Screen Identifies Compounds that Upregulate the p53 Isoform Δ133p53α and Inhibit Cellular Senescence.

定量高通量筛选鉴定出能上调 p53 同工型 Δ133p53α 并抑制细胞衰老的化合物

Lissa Delphine, Joruiz Sebastien M, Dranchak Patricia K, Ungerleider Kyra, Yamada Leo, Horikawa Izumi, Oliphant Erin, Manubag Rebecca, Von Muhlinen Natalia, Beck Jessica, Harris Brent T, Inglese James, Harris Curtis

Uncovering the isoform-resolution kinetic landscape of nonsense-mediated mRNA decay with EZbakR

利用 EZbakR 揭示无义介导的 mRNA 衰变的异构体分辨率动力学图谱

Mabin, Justin W; Vock, Isaac W; Machyna, Martin; Haque, Nazmul; Thakran, Poonam; Zhang, Alexandra; Rai, Ganesha; Leibler, Isabelle Nathalie-Marie; Inglese, James; Simon, Matthew D; Hogg, J Robert

Pharmacologic activation of Δ133p53α reduces cellular senescence in progeria patients-derived cells

药物激活Δ133p53α可减少早衰症患者来源细胞的衰老

Joruiz, Sebastien M; Lissa, Delphine; Von Muhlinen, Natalia; Dranchak, Patricia K; Inglese, James; Horikawa, Izumi; Harris, Curtis C

A Differential Ion Mobility Acoustic Ejection Mass Spectrometer System for Screening Isomerization-Mediating Enzyme Drug Targets

用于筛选异构化介导酶药物靶点的差分离子迁移率声波喷射质谱仪系统

Bazargan, Samad; Dranchak, Patricia; Liu, Chang; Inglese, James; Janiszewski, John; Schneider, Bradley B; Covey, Thomas R

qHTSWaterfall: 3-dimensional visualization software for quantitative high-throughput screening (qHTS) data

qHTSWaterfall:用于定量高通量筛选 (qHTS) 数据的三维可视化软件

Queme, Bryan; Braisted, John C; Dranchak, Patricia; Inglese, James

The NCATS Assay Guidance Manual programme: advancing the practice and rigour of preclinical translation

NCATS检测指导手册计划:推进临床前转化实践和严谨性

Markossian, Sarine; Brimacombe, Kyle R; Sittampalam, G Sitta; Grossman, Abigail; Coussens, Nathan P; Inglese, James; Auld, Douglas S; Chin, William; Austin, Christopher P; Hall, Matthew D

Ipomoeassin F Binds Sec61α to Inhibit Protein Translocation

番薯素F与Sec61α结合以抑制蛋白质转位

Zong, Guanghui; Hu, Zhijian; O'Keefe, Sarah; Tranter, Dale; Iannotti, Michael J; Baron, Ludivine; Hall, Belinda; Corfield, Katherine; Paatero, Anja O; Henderson, Mark J; Roboti, Peristera; Zhou, Jianhong; Sun, Xianwei; Govindarajan, Mugunthan; Rohde, Jason M; Blanchard, Nicolas; Simmonds, Rachel; Inglese, James; Du, Yuchun; Demangel, Caroline; High, Stephen; Paavilainen, Ville O; Shi, Wei Q