日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Workflow for E3 Ligase Ligand Validation for PROTAC Development

PROTAC 开发中 E3 连接酶配体验证的工作流程

Miletić, Nebojša; Weckesser, Janik; Mosler, Thorsten; Rathore, Rajeshwari; Hoffmann, Marina E; Gehrtz, Paul; Schlesiger, Sarah; Hartung, Ingo V; Berner, Nicola; Wilhelm, Stephanie; Müller, Juliane; Adhikari, Bikash; Němec, Václav; Sivashanmugam, Saran Aswathaman; Elson, Lewis; Holzmann, Hanna; Schwalm, Martin P; Hoffmann, Lasse; Abdul Azeez, Kamal Rayees; Müller, Susanne; Kuster, Bernhard; Wolf, Elmar; Đikić, Ivan; Knapp, Stefan

Introduction to the themed collection on 'Induced-Proximity Pharmacology'

“诱导邻近药理学”主题系列介绍

Hartung, Ingo V; James, Lindsey I; Jones, Lyn H

Discovery of BAY-405: An Azaindole-Based MAP4K1 Inhibitor for the Enhancement of T-Cell Immunity against Cancer

BAY-405 的发现:一种基于氮杂吲哚的 MAP4K1 抑制剂,可增强 T 细胞对癌症的免疫力

Jeffrey Mowat ,Rafael Carretero ,Gabriele Leder ,Nuria Aiguabella Font ,Roland Neuhaus ,Sandra Berndt ,Judith Günther ,Anders Friberg ,Martina Schäfer ,Hans Briem ,Marian Raschke ,Hideki Miyatake Ondozabal ,Bernd Buchmann ,Ulf Boemer ,Bertolt Kreft ,Ingo V Hartung ,Rienk Offringa

A miniaturized mode-of-action profiling platform enables high throughput characterization of the molecular and cellular dynamics of EZH2 inhibition

微型作用模式分析平台能够高通量表征 EZH2 抑制的分子和细胞动力学

Lilia Falkenstern #, Victoria Georgi #, Stefanie Bunse, Volker Badock, Manfred Husemann, Ulrike Roehn, Timo Stellfeld, Mark Fitzgerald, Steven Ferrara, Detlef Stöckigt, Carlo Stresemann, Ingo V Hartung, Amaury Fernández-Montalván

Target 2035 - an update on private sector contributions

2035年目标——私营部门贡献的最新情况

Ackloo, Suzanne; Antolin, Albert A; Bartolome, Jose Manuel; Beck, Hartmut; Bullock, Alex; Betz, Ulrich A K; Böttcher, Jark; Brown, Peter J; Chaturvedi, Menorca; Crisp, Alisa; Daniels, Danette; Dreher, Jan; Edfeldt, Kristina; Edwards, Aled M; Egner, Ursula; Elkins, Jon; Fischer, Christian; Glendorf, Tine; Goldberg, Steven; Hartung, Ingo V; Hillisch, Alexander; Homan, Evert; Knapp, Stefan; Köster, Markus; Krämer, Oliver; Llaveria, Josep; Lessel, Uta; Lindemann, Sven; Linderoth, Lars; Matsui, Hisanori; Michel, Maurice; Montel, Florian; Mueller-Fahrnow, Anke; Müller, Susanne; Owen, Dafydd R; Saikatendu, Kumar Singh; Santhakumar, Vijayaratnam; Sanderson, Wendy; Scholten, Cora; Schapira, Matthieu; Sharma, Sujata; Shireman, Brock; Sundström, Michael; Todd, Matthew H; Tredup, Claudia; Venable, Jennifer; Willson, Timothy M; Arrowsmith, Cheryl H

Target 2035 - update on the quest for a probe for every protein

2035年目标——为每种蛋白质寻找探针的最新进展

Müller, Susanne; Ackloo, Suzanne; Al Chawaf, Arij; Al-Lazikani, Bissan; Antolin, Albert; Baell, Jonathan B; Beck, Hartmut; Beedie, Shaunna; Betz, Ulrich A K; Bezerra, Gustavo Arruda; Brennan, Paul E; Brown, David; Brown, Peter J; Bullock, Alex N; Carter, Adrian J; Chaikuad, Apirat; Chaineau, Mathilde; Ciulli, Alessio; Collins, Ian; Dreher, Jan; Drewry, David; Edfeldt, Kristina; Edwards, Aled M; Egner, Ursula; Frye, Stephen V; Fuchs, Stephen M; Hall, Matthew D; Hartung, Ingo V; Hillisch, Alexander; Hitchcock, Stephen H; Homan, Evert; Kannan, Natarajan; Kiefer, James R; Knapp, Stefan; Kostic, Milka; Kubicek, Stefan; Leach, Andrew R; Lindemann, Sven; Marsden, Brian D; Matsui, Hisanori; Meier, Jordan L; Merk, Daniel; Michel, Maurice; Morgan, Maxwell R; Mueller-Fahrnow, Anke; Owen, Dafydd R; Perry, Benjamin G; Rosenberg, Saul H; Saikatendu, Kumar Singh; Schapira, Matthieu; Scholten, Cora; Sharma, Sujata; Simeonov, Anton; Sundström, Michael; Superti-Furga, Giulio; Todd, Matthew H; Tredup, Claudia; Vedadi, Masoud; von Delft, Frank; Willson, Timothy M; Winter, Georg E; Workman, Paul; Arrowsmith, Cheryl H

Donated chemical probes for open science

捐赠化学探针用于开放科学

Müller, Susanne; Ackloo, Suzanne; Arrowsmith, Cheryl H; Bauser, Marcus; Baryza, Jeremy L; Blagg, Julian; Böttcher, Jark; Bountra, Chas; Brown, Peter J; Bunnage, Mark E; Carter, Adrian J; Damerell, David; Dötsch, Volker; Drewry, David H; Edwards, Aled M; Edwards, James; Elkins, Jon M; Fischer, Christian; Frye, Stephen V; Gollner, Andreas; Grimshaw, Charles E; IJzerman, Adriaan; Hanke, Thomas; Hartung, Ingo V; Hitchcock, Steve; Howe, Trevor; Hughes, Terry V; Laufer, Stefan; Li, Volkhart Mj; Liras, Spiros; Marsden, Brian D; Matsui, Hisanori; Mathias, John; O'Hagan, Ronan C; Owen, Dafydd R; Pande, Vineet; Rauh, Daniel; Rosenberg, Saul H; Roth, Bryan L; Schneider, Natalie S; Scholten, Cora; Singh Saikatendu, Kumar; Simeonov, Anton; Takizawa, Masayuki; Tse, Chris; Thompson, Paul R; Treiber, Daniel K; Viana, Amélia Yi; Wells, Carrow I; Willson, Timothy M; Zuercher, William J; Knapp, Stefan; Mueller-Fahrnow, Anke

Discovery of Molidustat (BAY 85-3934): A Small-Molecule Oral HIF-Prolyl Hydroxylase (HIF-PH) Inhibitor for the Treatment of Renal Anemia

莫利司他(BAY 85-3934)的发现:一种用于治疗肾性贫血的小分子口服HIF-脯氨酰羟化酶(HIF-PH)抑制剂

Beck, Hartmut; Jeske, Mario; Thede, Kai; Stoll, Friederike; Flamme, Ingo; Akbaba, Metin; Ergüden, Jens-Kerim; Karig, Gunter; Keldenich, Jörg; Oehme, Felix; Militzer, Hans-Christian; Hartung, Ingo V; Thuss, Uwe

Discovery and Characterization of a Highly Potent and Selective Aminopyrazoline-Based in Vivo Probe (BAY-598) for the Protein Lysine Methyltransferase SMYD2

发现并表征针对蛋白质赖氨酸甲基转移酶 SMYD2 的高效选择性氨基吡唑啉类体内探针 (BAY-598)

Erik Eggert, Roman C Hillig, Silke Koehr, Detlef Stöckigt, Jörg Weiske, Naomi Barak, Jeffrey Mowat, Thomas Brumby, Clara D Christ, Antonius Ter Laak, Tina Lang, Amaury E Fernandez-Montalvan, Volker Badock, Hilmar Weinmann, Ingo V Hartung, Dalia Barsyte-Lovejoy, Magdalena Szewczyk, Steven Kennedy, Fe