日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exploiting the 2-(1,3,4,9-tetrahydropyrano[3,4-b]indol-1-yl)acetic Acid Scaffold to Generate COXTRANs: A New Class of Dual Cyclooxygenase Inhibitors-Thromboxane Receptor Antagonists

利用 2-(1,3,4,9-四氢吡喃并[3,4-b]吲哚-1-基)乙酸骨架生成 COXTRANs:一类新型双重环氧合酶抑制剂-血栓素受体拮抗剂

Blua, Federica; Boccato, Francesca; Buccellati, Carola; Risè, Patrizia; Barbieri, Silvia; Castiglioni, Laura; Balzulat, Annika; Rolando, Barbara; Marini, Elisabetta; Balestra, Marta; Introvigne, Maria Luisa; Giorgis, Marta; Sironi, Luigi; Tacconelli, Stefania; Hiesinger, Kerstin; Patrignani, Paola; Schmidtko, Achim; Steinhilber, Dieter; Proschak, Ewgenij; Sala, Angelo; Rovati, G Enrico; Bertinaria, Massimo

Restoring cefepime activity against multidrug-resistant KPC-producing Klebsiella pneumoniae by combination with boronic acid inhibitors, MB076 and S02030

通过与硼酸抑制剂 MB076 和 S02030 联合使用,恢复头孢吡肟对多重耐药性产 KPC 肺炎克雷伯菌的活性

Rojas, Laura J; Nielsen, Travis B; Pantapalangkoor, Paul; Taracila, Magdalena A; Introvigne, Maria L; Sharma, Rajnikant; Yeshwante, Shekhar; Mojica, Maria F; Papp-Wallace, Krisztina M; Hujer, Andrea M; Prati, Fabio; Caselli, Emilia; Spellberg, Brad; Rather, Philip N; Rao, Gauri G; Bonomo, Robert A

α-Triazolylboronic Acids: A Novel Scaffold to Target FLT3 in AML

α-三唑基硼酸:一种靶向急性髓系白血病中FLT3的新型支架

Introvigne, Maria Luisa; Destro, Lorenza; Mologni, Luca; Crippa, Valentina; Zardi, Paolo; Fini, Francesco; Prati, Fabio; Caselli, Emilia; Zambon, Alfonso

Sulfonamidoboronic Acids as "Cross-Class" Inhibitors of an Expanded-Spectrum Class C Cephalosporinase, ADC-33, and a Class D Carbapenemase, OXA-24/40: Strategic Compound Design to Combat Resistance in Acinetobacter baumannii

磺酰胺硼酸作为广谱C类头孢菌素酶ADC-33和D类碳青霉烯酶OXA-24/40的“跨类别”抑制剂:对抗鲍曼不动杆菌耐药性的策略性化合物设计

Introvigne, Maria Luisa; Beardsley, Trevor J; Fernando, Micah C; Leonard, David A; Wallar, Bradley J; Rudin, Susan D; Taracila, Magdalena A; Rather, Philip N; Colquhoun, Jennifer M; Song, Shaina; Fini, Francesco; Hujer, Kristine M; Hujer, Andrea M; Prati, Fabio; Powers, Rachel A; Bonomo, Robert A; Caselli, Emilia

Boronic Acid Transition State Inhibitors as Potent Inactivators of KPC and CTX-M β-Lactamases: Biochemical and Structural Analyses

硼酸过渡态抑制剂作为 KPC 和 CTX-M β-内酰胺酶的强效灭活剂:生化和结构分析

Tahani A Alsenani, María Margarita Rodríguez, Barbara Ghiglione, Magdalena A Taracila, Maria F Mojica, Laura J Rojas, Andrea M Hujer, Gabriel Gutkind, Christopher R Bethel, Philip N Rather, Maria Luisa Introvigne, Fabio Prati, Emilia Caselli, Pablo Power, Focco van den Akker, Robert A Bonomo3

α-Triazolylboronic Acids: A Promising Scaffold for Effective Inhibitors of KPCs

α-三唑基硼酸:一种有前景的KPC有效抑制剂骨架

Introvigne, Maria Luisa; Taracila, Magdalena A; Prati, Fabio; Caselli, Emilia; Bonomo, Robert A