日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Polyfunctionalized N-Arylsulfonyl Indoles: Identification of (E)-N-Hydroxy-3-{3-[(5-(3-(piperidin-1-yl)propoxy]-1H-indol-1-yl)sulfonyl]phenyl}acrylamide (MTP150) for the Epigenetic-Based Therapy of Parkinson's Disease

多功能化N-芳基磺酰基吲哚:(E)-N-羟基-3-{3-[(5-(3-(哌啶-1-基)丙氧基]-1H-吲哚-1-基)磺酰基]苯基}丙烯酰胺 (MTP150) 的鉴定及其在帕金森病表观遗传治疗中的应用

Toledano-Pinedo, Mireia; Porro-Pérez, Alicia; Schäker-Hübner, Linda; Diez-Iriepa, Daniel; Iriepa, Isabel; Siwek, Agata; Wolak, Małgorzata; Satała, Grzegorz; Bojarski, Andrzej J; Doroz-Płonka, Agata; Handzlik, Jadwiga; Godyń, Justyna; Dallemagne, Patrick; Rochais, Christophe; Davis, Audrey; Since, Marc; Pérez, Belén; Bellver-Sanchis, Aina; Irisarri, Alba; Pallàs, Mercè; Solana-Manrique, Cristina; López-Muñoz, Francisco; Ismaili, Lhassane; Griñán-Ferré, Christian; Paricio, Nuria; K Hansen, Finn; Więckowska, Anna; Marco-Contelles, José

Generation and validation of a novel multitarget small molecule in glioblastoma.

胶质母细胞瘤新型多靶点小分子的生成与验证

Artetxe-Zurutuza Aizpea, Iturrioz-Rodriguez Nerea, Elizazu Joseba, Toledano-Pinedo Mireia, Porro-Pérez Alicia, De Goñi Irati, Elua-Pinin Alejandro, Schäker-Hübner Linda, Azkargorta Mikel, Elortza Felix, Iriepa Isabel, Lòpez-Muñoz Francisco, Moncho-Amor Veronica, Hansen Finn K, Sampron Nicolás, Marco-Contelles Jose Luis, Matheu Ander

Designing Molecular Solar Thermal Systems Based on the Paternò-Büchi Reaction Coupled to Enzymatic Energy Release

基于Paternò-Büchi反应耦合酶促能量释放的分子太阳能热系统设计

Delgado-Gómez, Marta; Reategui Illatopa, Jesús; Gramolini, Lorenzo; López-Corbalán, Richard; García-Iriepa, Cristina; Marazzi, Marco

Coinage Metal-Catalyzed Divergent Heterocyclizations of Underexplored N-Propargyl Hydrazides

贵金属催化的未充分研究的N-炔丙基酰肼的发散性杂环化反应

Diez-Iriepa, Daniel; Toledano-Pinedo, Mireia; Herrera-Hernández, Lorena; Samadi, Abdelouahid; Raouf, Yasir S; Rodríguez-Fernández, M Mercedes; Flores-Galán, Paula; Yanai, Hikaru; Alonso, José M; Marco-Contelles, José; Almendros, Pedro

Multicomponent Synthesis of Multi-Target Quinazolines Modulating Cholinesterase, Oxidative Stress, and Amyloid Aggregation Activities for the Therapy of Alzheimer's Disease

利用多组分合成法制备多靶点喹唑啉类化合物,调节胆碱酯酶、氧化应激和淀粉样蛋白聚集活性,用于治疗阿尔茨海默病

Chakhari, Saida; Marco-Contelles, José; Iriepa, Isabel; Carreiras, Maria do Carmo; Chabchoub, Fakher; Ismaili, Lhassane; Refouvelet, Bernard

Modulating Efficiency and Color of Thermally Activated Delayed Fluorescence by Rationalizing the Substitution Effect

通过合理化取代效应来调控热激活延迟荧光的效率和颜色

Jodra, Alejandro; Marazzi, Marco; Frutos, Luis Manuel; García-Iriepa, Cristina

8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseases

8-羟基喹啉基硝酮作为治疗神经退行性疾病的多功能配体

Knez, Damijan; Diez-Iriepa, Daniel; Chioua, Mourad; Gottinger, Andrea; Denic, Milica; Chantegreil, Fabien; Nachon, Florian; Brazzolotto, Xavier; Skrzypczak-Wiercioch, Anna; Meden, Anže; Pišlar, Anja; Kos, Janko; Žakelj, Simon; Stojan, Jure; Sałat, Kinga; Serrano, Julia; Fernández, Ana Patricia; Sánchez-García, Aitana; Martínez-Murillo, Ricardo; Binda, Claudia; López-Muñoz, Francisco; Gobec, Stanislav; Marco-Contelles, José

An Algorithm Predicting the Optimal Mechanical Response of Electronic Energy Difference

一种预测电子能量差最优机械响应的算法

Jodra, Alejandro; García-Iriepa, Cristina; Frutos, Luis Manuel

Straightforward Synthesis of Bis[(trifluoromethyl)sulfonyl]ethylated Isocoumarins from 2-Ethynylbenzoates

由2-乙炔基苯甲酸酯直接合成双[(三氟甲基)磺酰基]乙基化异香豆素

Petcu, A Sonia; Lázaro-Milla, Carlos; Rodríguez, F Javier; Iriepa, Isabel; Bautista-Aguilera, Óscar M; Aragoncillo, Cristina; Alonso, José M; Almendros, Pedro

Polyfunctionalized α-Phenyl-tert-butyl(benzyl)nitrones: Multifunctional Antioxidants for Stroke Treatment

多功能化α-苯基叔丁基(苄基)硝酮:用于中风治疗的多功能抗氧化剂

Diez-Iriepa, Daniel; Knez, Damijan; Gobec, Stanislav; Iriepa, Isabel; de Los Ríos, Cristóbal; Bravo, Isaac; López-Muñoz, Francisco; Marco-Contelles, José; Hadjipavlou-Litina, Dimitra