日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Polyfunctionalized N-Arylsulfonyl Indoles: Identification of (E)-N-Hydroxy-3-{3-[(5-(3-(piperidin-1-yl)propoxy]-1H-indol-1-yl)sulfonyl]phenyl}acrylamide (MTP150) for the Epigenetic-Based Therapy of Parkinson's Disease

多功能化N-芳基磺酰基吲哚:(E)-N-羟基-3-{3-[(5-(3-(哌啶-1-基)丙氧基]-1H-吲哚-1-基)磺酰基]苯基}丙烯酰胺 (MTP150) 的鉴定及其在帕金森病表观遗传治疗中的应用

Toledano-Pinedo, Mireia; Porro-Pérez, Alicia; Schäker-Hübner, Linda; Diez-Iriepa, Daniel; Iriepa, Isabel; Siwek, Agata; Wolak, Małgorzata; Satała, Grzegorz; Bojarski, Andrzej J; Doroz-Płonka, Agata; Handzlik, Jadwiga; Godyń, Justyna; Dallemagne, Patrick; Rochais, Christophe; Davis, Audrey; Since, Marc; Pérez, Belén; Bellver-Sanchis, Aina; Irisarri, Alba; Pallàs, Mercè; Solana-Manrique, Cristina; López-Muñoz, Francisco; Ismaili, Lhassane; Griñán-Ferré, Christian; Paricio, Nuria; K Hansen, Finn; Więckowska, Anna; Marco-Contelles, José

Masupirdine, a Selective Serotonin 5‑HT(6) Receptor Antagonist for Alzheimer's Disease

马苏匹啶,一种用于治疗阿尔茨海默病的选择性5-羟色胺5-HT(6)受体拮抗剂

Toledano-Pinedo, Mireia; Iriepa, Isabel; Rodríguez-Fernández, M Mercedes; Marco-Contelles, José

Generation and validation of a novel multitarget small molecule in glioblastoma.

胶质母细胞瘤新型多靶点小分子的生成与验证

Artetxe-Zurutuza Aizpea, Iturrioz-Rodriguez Nerea, Elizazu Joseba, Toledano-Pinedo Mireia, Porro-Pérez Alicia, De Goñi Irati, Elua-Pinin Alejandro, Schäker-Hübner Linda, Azkargorta Mikel, Elortza Felix, Iriepa Isabel, Lòpez-Muñoz Francisco, Moncho-Amor Veronica, Hansen Finn K, Sampron Nicolás, Marco-Contelles Jose Luis, Matheu Ander

2-{N-[ω-(1-Benzylpiperidin-4-yl)alkyl]amino}-6-[(prop-2-yn-1-yl)amino]pyridine-3,5-dicarbonitriles Showing High Affinity for σ(1/2) Receptors

2-{N-[ω-(1-苄基哌啶-4-基)烷基]氨基}-6-[(丙-2-炔-1-基)氨基]吡啶-3,5-二腈对σ(1/2)受体表现出高亲和力

Deuther-Conrad, Winnie; Schepmann, Dirk; Iriepa, Isabel; López-Muñoz, Francisco; Chioua, Mourad; Wünsch, Bernhard; Samadi, Abdelouahid; Marco-Contelles, José

Piperidine-catalyzed synthesis of (E)-2-cyanoacrylamides: crystallographic, antiproliferative, and docking studies

哌啶催化合成(E)-2-氰基丙烯酰胺:晶体学、抗增殖和分子对接研究

Serrano-Sterling, Camilo; Iriepa, Isabel; Macías, Mario A; Castillo, Juan-Carlos; Becerra, Diana

Multicomponent Synthesis of Multi-Target Quinazolines Modulating Cholinesterase, Oxidative Stress, and Amyloid Aggregation Activities for the Therapy of Alzheimer's Disease

利用多组分合成法制备多靶点喹唑啉类化合物,调节胆碱酯酶、氧化应激和淀粉样蛋白聚集活性,用于治疗阿尔茨海默病

Chakhari, Saida; Marco-Contelles, José; Iriepa, Isabel; Carreiras, Maria do Carmo; Chabchoub, Fakher; Ismaili, Lhassane; Refouvelet, Bernard

Zervimesine, a Small Sigma‑2 Receptor Selective Modulator for Alzheimer's Disease

泽维美辛,一种用于治疗阿尔茨海默病的选择性小分子σ-2受体调节剂

Iriepa, Isabel; Contino, Marialessandra; Abate, Carmen; Marco-Contelles, José

Straightforward Synthesis of Bis[(trifluoromethyl)sulfonyl]ethylated Isocoumarins from 2-Ethynylbenzoates

由2-乙炔基苯甲酸酯直接合成双[(三氟甲基)磺酰基]乙基化异香豆素

Petcu, A Sonia; Lázaro-Milla, Carlos; Rodríguez, F Javier; Iriepa, Isabel; Bautista-Aguilera, Óscar M; Aragoncillo, Cristina; Alonso, José M; Almendros, Pedro

Polyfunctionalized α-Phenyl-tert-butyl(benzyl)nitrones: Multifunctional Antioxidants for Stroke Treatment

多功能化α-苯基叔丁基(苄基)硝酮:用于中风治疗的多功能抗氧化剂

Diez-Iriepa, Daniel; Knez, Damijan; Gobec, Stanislav; Iriepa, Isabel; de Los Ríos, Cristóbal; Bravo, Isaac; López-Muñoz, Francisco; Marco-Contelles, José; Hadjipavlou-Litina, Dimitra

Homo-Tris-Nitrones Derived from α-Phenyl-N-tert-butylnitrone: Synthesis, Neuroprotection and Antioxidant Properties

α-苯基-N-叔丁基硝酮衍生的同型三硝酮:合成、神经保护和抗氧化特性

Diez-Iriepa, Daniel; Chamorro, Beatriz; Talaván, Marta; Chioua, Mourad; Iriepa, Isabel; Hadjipavlou-Litina, Dimitra; López-Muñoz, Francisco; Marco-Contelles, José; Oset-Gasque, María Jesús