日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The ATC12 small molecule inhibits the Aurora-A/TPX2 interaction and impairs the proliferation of breast cancer cells

ATC12小分子抑制Aurora-A/TPX2相互作用,从而抑制乳腺癌细胞增殖。

Boi, Dalila; Fianco, Giulia; Polverino, Federica; Fiorentino, Francesco; Mastrangelo, Anna; Rossi, Simone; Rubini, Elisabetta; Rosignoli, Serena; Troilo, Francesca; Antonelli, Maria Rosaria; Tarquini, Dalila; Cervoni, Laura; Rinaldo, Serena; Tramonti, Angela; Scarpone, Eleonora Kristina; Naro, Chiara; Sette, Claudio; Stagni, Venturina; Colotti, Gianni; Rotili, Dante; Paiardini, Alessandro; Guarguaglini, Giulia; Asteriti, Italia Anna

AurkA nuclear localization is promoted by TPX2 and counteracted by protein degradation

TPX2 促进 AurkA 核定位,并被蛋白质降解所抵消

Italia Anna Asteriti, Federica Polverino, Venturina Stagni, Valentina Sterbini, Camilla Ascanelli, Francesco Davide Naso, Anna Mastrangelo, Alessandro Rosa, Alessandro Paiardini, Catherine Lindon, Giulia Guarguaglini

AurkA nuclear localization is promoted by TPX2 and counteracted by protein degradation

TPX2促进AurkA的核定位,而蛋白质降解则抑制AurkA的核定位。

Italia Anna Asteriti,Federica Polverino,Venturina Stagni,Valentina Sterbini,Camilla Ascanelli,Francesco Davide Naso,Anna Mastrangelo,Alessandro Rosa,Alessandro Paiardini,Catherine Lindon,Giulia Guarguaglini

Revisiting degron motifs in human AURKA required for its targeting by APC/CFZR1

重新审视人类 AURKA 中 APC/CFZR1 靶向所需的降解基序

Ahmed Abdelbaki, Camilla Ascanelli, Cynthia N Okoye, H Begum Akman, Giacomo Janson, Mingwei Min, Chiara Marcozzi, Anja Hagting, Rhys Grant, Maria De Luca, Italia Anna Asteriti, Giulia Guarguaglini, Alessandro Paiardini, Catherine Lindon

Visualization of human karyopherin beta-1/importin beta-1 interactions with protein partners in mitotic cells by co-immunoprecipitation and proximity ligation assays

通过共免疫沉淀和邻近连接试验可视化人类核转运蛋白β-1/输入蛋白β-1与有丝分裂细胞中的蛋白质伙伴的相互作用

Laura Di Francesco, Annalisa Verrico, Italia Anna Asteriti, Paola Rovella, Pietro Cirigliano, Giulia Guarguaglini, Maria Eugenia Schininà, Patrizia Lavia

Identification of small molecule inhibitors of the Aurora-A/TPX2 complex

Aurora-A/TPX2复合物小分子抑制剂的鉴定

Italia Anna Asteriti, Frederick Daidone, Gianni Colotti, Serena Rinaldo, Patrizia Lavia, Giulia Guarguaglini, Alessandro Paiardini

Subcellular localization of the five members of the human steroid 5α-reductase family

人类类固醇 5α-还原酶家族五个成员的亚细胞定位

Antonella Scaglione, Linda Celeste Montemiglio, Giacomo Parisi, Italia Anna Asteriti, Renato Bruni, Gabriele Cerutti, Claudia Testi, Carmelinda Savino, Filippo Mancia, Patrizia Lavia, Beatrice Vallone

Cross-Talk between AURKA and Plk1 in Mitotic Entry and Spindle Assembly

AURKA 和 Plk1 在有丝分裂起始和纺锤体组装中的相互作用

Asteriti, Italia Anna; De Mattia, Fabiola; Guarguaglini, Giulia

The Aurora-A inhibitor MLN8237 affects multiple mitotic processes and induces dose-dependent mitotic abnormalities and aneuploidy

Aurora-A 抑制剂 MLN8237 影响多种有丝分裂过程,并诱导剂量依赖性的有丝分裂异常和非整倍性

Italia Anna Asteriti, Erica Di Cesare, Fabiola De Mattia, Volker Hilsenstein, Beate Neumann, Enrico Cundari, Patrizia Lavia, Giulia Guarguaglini