日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

RNA-binding protein LARP6 coordinates hepatic stellate cell activation and liver fibrosis

RNA结合蛋白LARP6协调肝星状细胞活化和肝纤维化

Kim, Hyun Young; Mizrahi, Orel; Lee, Wonseok; Rosenthal, Sara B; Han, Cuijuan; Yee, Brian A; Blue, Steven M; Diaz, Jesiel; Jonnalagadda, Jyotiprakash P; Street, Lena A; Hokutan, Kanani; Jang, Haeum; Miciano, Charlene; Ma, Chen-Ting; Bobkov, Andrey A; Sergienko, Eduard; Jackson, Michael R; Jovanovic, Marko; Stefanovic, Branko; Kisseleva, Tatiana; Yeo, Gene W; Brenner, David A

Designing allosteric modulators to change GPCR G protein subtype selectivity

设计变构调节剂以改变GPCR G蛋白亚型选择性

Moore, Madelyn N; Person, Kelsey L; Robleto, Valeria L; Alwin, Abigail R; Krusemark, Campbell L; Foster, Noah; Ray, Caroline; Inoue, Asuka; Jackson, Michael R; Sheedlo, Michael J; Barak, Lawrence S; Marron Fernandez de Velasco, Ezequiel; Olson, Steven H; Slosky, Lauren M

Arrestin-biased allosteric modulator of neurotensin receptor 1 alleviates acute and chronic pain.

神经降压素受体 1 的 Arrestin 偏向性变构调节剂可缓解急性和慢性疼痛

Guo Ran, Chen Ouyang, Zhou Yang, Bang Sangsu, Chandra Sharat, Li Yize, Chen Gang, Xie Rou-Gang, He Wei, Xu Jing, Zhou Richard, Song Shaoyong, Person Kelsey L, Moore Madelyn N, Alwin Abigail R, Spasojevic Ivan, Jackson Michael R, Olson Steven H, Caron Marc G, Slosky Lauren M, Wetsel William C, Barak Lawrence S, Ji Ru-Rong

GPR25 promotes the formation of lung and liver tissue-resident memory CD8 T cells

GPR25促进肺和肝组织驻留记忆CD8 T细胞的形成

Feng, Han; Park, Sungjun; Shin, Jae Woo; Castañeda-Castro, Francisco Emmanuel; Hernandez, Job Rocha; Schmiedel, Benjamin J; Liu, Changlu; Jackson, Michael R; Ottensmeier, Christian H; Vijayanand, Pandurangan

Biased allosteric modulator of neurotensin receptor 1 reduces ethanol drinking and responses to ethanol administration in rodents

神经降压素受体1的偏向性变构调节剂可降低啮齿动物的乙醇摄入量和对乙醇给药的反应

Gereau, Graydon B; Zhou, Diana; Voorhies, Kalynn Van; Tyler, Ryan E; Campbell, Jeffrey; Murray, Jackson G; Alvarez-Pamir, Ali; Wykoff, Luke A; Companion, Michel A; Jackson, Michael R; Olson, Steven H; Barak, Lawrence S; Slosky, Lauren M; Vetreno, Ryan P; Besheer, Joyce; McElligott, Zoe A

β-arrestin-biased Allosteric Modulator of Neurotensin Receptor 1 Reduces Ethanol Drinking and Responses to Ethanol Administration in Rodents

β-arrestin偏向性神经降压素受体1变构调节剂可降低啮齿动物的乙醇摄入量和对乙醇给药的反应

Gereau, Graydon B; Zhou, Diana; Van Voorhies, Kalynn; Tyler, Ryan E; Campbell, Jeffrey; Murray, Jackson G; Alvarez-Pamir, Ali; Wykoff, Luke A; Companion, Michel A; Jackson, Michael R; Olson, Steven H; Barak, Lawrence S; Slosky, Lauren M; Vetreno, Ryan P; Besheer, Joyce; McElligott, Zoe A

Discovery of a first-in-class inhibitor of sulfide:quinone oxidoreductase that protects against adverse cardiac remodelling and heart failure

发现一种首创的硫化物:醌氧化还原酶抑制剂,可预防不良心脏重塑和心力衰竭

Jackson, Michael R; Cox, Kristie D; Baugh, Simon D P; Wakeen, Luke; Rashad, Adel A; Lam, Patrick Y S; Polyak, Boris; Jorns, Marilyn Schuman

Synthesis and evaluation of potent novel inhibitors of human sulfide:quinone oxidoreductase

合成和评价新型高效人硫化物:醌氧化还原酶抑制剂

Baugh, Simon D P; Jackson, Michael R; Rashad, Adel Ahmed; Reitz, Allen B; Lam, Patrick Y S; Jorns, Marilyn Schuman

Discovery of 5-((5-chloro-2-methoxyphenyl)sulfonamido)nicotinamide (SBI-425), a potent and orally bioavailable tissue-nonspecific alkaline phosphatase (TNAP) inhibitor

发现 5-((5-氯-2-甲氧基苯基)磺酰胺基)烟酰胺 (SBI-425),一种强效且口服生物利用度高的组织非特异性碱性磷酸酶 (TNAP) 抑制剂

Pinkerton, Anthony B; Sergienko, Eduard; Bravo, Yalda; Dahl, Russell; Ma, Chen-Ting; Sun, Qing; Jackson, Michael R; Cosford, Nicholas D P; Millán, José Luis

Signal transduction controls heterogeneous NF-κB dynamics and target gene expression through cytokine-specific refractory states

信号转导通过细胞因子特异性不应期控制异质性 NF-κB 动力学和靶基因表达

Antony Adamson, Christopher Boddington, Polly Downton, William Rowe, James Bagnall, Connie Lam, Apolinar Maya-Mendoza, Lorraine Schmidt, Claire V Harper, David G Spiller, David A Rand, Dean A Jackson, Michael R H White, Pawel Paszek