Identification of Diarylurea Inhibitors of the Cardiac-Specific Kinase TNNI3K by Designing Selectivity Against VEGFR2, p38α, and B-Raf
通过设计针对 VEGFR2、p38α 和 B-Raf 的选择性来鉴定心脏特异性激酶 TNNI3K 的二芳脲抑制剂
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c00700
Jaclyn R Patterson, Alan P Graves, Patrick Stoy, Mui Cheung, Tina A Desai, Harvey Fries, Gregory J Gatto Jr, Dennis A Holt, Lisa Shewchuk, Rachel Totoritis, Liping Wang, Lara S Kallander